TargetHistamine H3 receptor(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Binding affinity to human H3 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity to rat H3 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Binding affinity to human H3 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Binding affinity to human H3 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 137nMAssay Description:Binding affinity to human recombinant DATMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 204nMAssay Description:Binding affinity to human recombinant M3 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 336nMAssay Description:Binding affinity to human recombinant M5 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 351nMAssay Description:Binding affinity to human recombinant M4 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 415nMAssay Description:Binding affinity to human recombinant M4 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 432nMAssay Description:Binding affinity to human recombinant 5HT1A receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 437nMAssay Description:Binding affinity to human recombinant M5 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 462nMAssay Description:Binding affinity to human recombinant M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 512nMAssay Description:Binding affinity to human recombinant M3 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 681nMAssay Description:Binding affinity to human recombinant M2 receptorMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 923nMAssay Description:Binding affinity to human recombinant H2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 931nMAssay Description:Binding affinity to human recombinant M1 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 1.36E+3nMAssay Description:Binding affinity to human recombinant 5HT2A receptorMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 1.71E+3nMAssay Description:Binding affinity to human recombinant H2 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 2.72E+3nMAssay Description:Binding affinity to human recombinant 5HT2A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 3.15E+3nMAssay Description:Binding affinity to human recombinant 5HT2B receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 3.27E+3nMAssay Description:Binding affinity to human recombinant M1 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 5.24E+3nMAssay Description:Binding affinity to human recombinant 5HT1D receptorMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 5.44E+3nMAssay Description:Binding affinity to human recombinant H1 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 6.38E+3nMAssay Description:Binding affinity to human recombinant 5HT1D receptorMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 7.06E+3nMAssay Description:Binding affinity to human recombinant H1 receptorMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant alpha2B adrenergic receptorMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant beta2 adrenergic receptorMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant beta2 adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant alpha2B adrenergic receptorMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant NETMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant SERTMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant NETMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT1B receptorMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant alpha1D adrenergic receptorMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant Dopamine D4 receptorMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant H4 receptorMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant H4 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT1B receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT2B receptorMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant DATMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT1E receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT1E receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT2C receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT2C receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT3 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT3 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT5A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT5A receptorMore data for this Ligand-Target Pair