Affinity DataKi: 164nMAssay Description:Binding affinity to 5HT2B receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataKi: 392nMAssay Description:Binding affinity to Sigma1More data for this Ligand-Target Pair
Affinity DataKi: 863nMAssay Description:Binding affinity to alpha1 adrenoreceptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 12.6nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 47.5nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 59.6nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 61.5nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 64.5nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 78.3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 80.8nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 92.5nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 93.8nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 97.6nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 139nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 149nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 164nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 174nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 264nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 289nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 369nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 434nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 452nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 495nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 502nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 534nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 660nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 772nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.02E+3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.07E+3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.28E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.86E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.98E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 2.05E+3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 2.11E+3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 5.77E+3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+3nMAssay Description:Antagonist activity at 5HT2A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 5.85E+3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 6.57E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 7.22E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 8.82E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.05E+4nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 5.25E+4nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals
Curated by ChEMBL
Sk Biopharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair