Compile Data Set for Download or QSAR
maximum 50k data
Found 46 Enz. Inhib. hit(s) with all data for entry = 50040401
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393649(CHEMBL2158704)
Affinity DataKi:  164nMAssay Description:Binding affinity to 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393649(CHEMBL2158704)
Affinity DataKi:  392nMAssay Description:Binding affinity to Sigma1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393649(CHEMBL2158704)
Affinity DataKi:  863nMAssay Description:Binding affinity to alpha1 adrenoreceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393658(CHEMBL2158721 | US8815852, 39)
Affinity DataIC50:  12.6nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393665(CHEMBL2158794)
Affinity DataIC50:  47.5nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393657(CHEMBL2158722)
Affinity DataIC50:  59.6nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393659(CHEMBL2158720 | US8815852, 36)
Affinity DataIC50:  61.5nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393651(CHEMBL2158705)
Affinity DataIC50:  62nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393655(CHEMBL2158725 | US8815852, 21)
Affinity DataIC50:  64.5nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393662(CHEMBL2158717)
Affinity DataIC50:  78.3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393660(CHEMBL2158719 | US8815852, 26)
Affinity DataIC50:  80.8nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393657(CHEMBL2158722)
Affinity DataIC50:  92.5nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393659(CHEMBL2158720 | US8815852, 36)
Affinity DataIC50:  93.8nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393661(CHEMBL2158718 | US8815852, 27)
Affinity DataIC50:  97.6nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393663(CHEMBL2158716 | US8815852, 41)
Affinity DataIC50:  110nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393650(CHEMBL2158706)
Affinity DataIC50:  139nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393662(CHEMBL2158717)
Affinity DataIC50:  149nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393663(CHEMBL2158716 | US8815852, 41)
Affinity DataIC50:  160nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393661(CHEMBL2158718 | US8815852, 27)
Affinity DataIC50:  164nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393667(CHEMBL2158795)
Affinity DataIC50:  174nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393654(CHEMBL2158726 | US8815852, 22)
Affinity DataIC50:  264nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393666(CHEMBL2158796)
Affinity DataIC50:  289nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393652(CHEMBL2158728)
Affinity DataIC50:  369nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393650(CHEMBL2158706)
Affinity DataIC50:  434nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393667(CHEMBL2158795)
Affinity DataIC50:  452nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393666(CHEMBL2158796)
Affinity DataIC50:  495nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393660(CHEMBL2158719 | US8815852, 26)
Affinity DataIC50:  502nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393651(CHEMBL2158705)
Affinity DataIC50:  534nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393658(CHEMBL2158721 | US8815852, 39)
Affinity DataIC50:  660nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393650(CHEMBL2158706)
Affinity DataIC50:  772nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393650(CHEMBL2158706)
Affinity DataIC50:  1.02E+3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393665(CHEMBL2158794)
Affinity DataIC50:  1.07E+3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393652(CHEMBL2158728)
Affinity DataIC50:  1.28E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393654(CHEMBL2158726 | US8815852, 22)
Affinity DataIC50:  1.86E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393649(CHEMBL2158704)
Affinity DataIC50:  1.98E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393656(CHEMBL2158723 | US8815852, 16)
Affinity DataIC50:  2.05E+3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393653(CHEMBL2158727)
Affinity DataIC50:  2.11E+3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393649(CHEMBL2158704)
Affinity DataIC50:  5.77E+3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393649(CHEMBL2158704)
Affinity DataIC50:  5.80E+3nMAssay Description:Antagonist activity at 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393649(CHEMBL2158704)
Affinity DataIC50:  5.85E+3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393656(CHEMBL2158723 | US8815852, 16)
Affinity DataIC50:  6.57E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393653(CHEMBL2158727)
Affinity DataIC50:  7.22E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393649(CHEMBL2158704)
Affinity DataIC50:  8.82E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393655(CHEMBL2158725 | US8815852, 21)
Affinity DataIC50:  1.05E+4nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393664(CHEMBL2158715)
Affinity DataIC50:  5.25E+4nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393664(CHEMBL2158715)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed