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Found 17 Enz. Inhib. hit(s) with all data for entry = 50039566
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50380097(CHEMBL2012935)
Affinity DataKi:  3.90E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50300802(5-Morpholin-4-ylpentanoic acid(4-pyridin-3-ylpheny...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50380100(CHEMBL2012937)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50380098(CHEMBL2010825)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50380099(CHEMBL2012936)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50380100(CHEMBL2012937)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50380098(CHEMBL2010825)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50380099(CHEMBL2012936)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50380097(CHEMBL2012935)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50300802(5-Morpholin-4-ylpentanoic acid(4-pyridin-3-ylpheny...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50380097(CHEMBL2012935)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50380100(CHEMBL2012937)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50380099(CHEMBL2012936)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50380098(CHEMBL2010825)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50300802(5-Morpholin-4-ylpentanoic acid(4-pyridin-3-ylpheny...)
Affinity DataEC50:  9.50E+3nMAssay Description:Partial agonist activity at wild type rat recombinant alpha7 nAChR expressed in Xenopus oocyte by voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50300811(CHEMBL576234 | N-{4-[4-(2,4-dimethoxyphenyl)-piper...)
Affinity DataEC50:  2.84E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50300802(5-Morpholin-4-ylpentanoic acid(4-pyridin-3-ylpheny...)
Affinity DataEC50:  1.65E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed