Compile Data Set for Download or QSAR
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Found 12 Enz. Inhib. hit(s) with all data for entry = 50040970
TargetToll-like receptor 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403022(CHEMBL2216760)
Affinity DataEC50:  4.13E+4nMAssay Description:Agonist activity at human TLR8 transfected in HEK cells assessed as NFkappaB induction after 24 hrs by specific secreted alkaline phosphatase gene as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403023(CHEMBL2216759)
Affinity DataEC50: >2.70E+5nMAssay Description:Agonist activity at human TLR8 transfected in HEK cells assessed as NFkappaB induction after 24 hrs by specific secreted alkaline phosphatase gene as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50320082(1-(4-Amino-2-butyl-1H-imidazo-[4,5-c]quinolin-1-yl...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human TLR8 transfected in HEK cells assessed as NFkappaB induction after 24 hrs by specific secreted alkaline phosphatase gene as...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403024(CHEMBL195276)
Affinity DataEC50: >2.70E+5nMAssay Description:Agonist activity at human TLR8 transfected in HEK cells assessed as NFkappaB induction after 24 hrs by specific secreted alkaline phosphatase gene as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50241029(1-[4-amino-2-(ethoxymethyl)-1H-imidazo[4,5-c]quino...)
Affinity DataEC50:  6.40E+3nMAssay Description:Agonist activity at human TLR8 transfected in HEK cells assessed as NFkappaB induction after 24 hrs by specific secreted alkaline phosphatase gene as...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50240849(1-(2-methylpropyl)-1H-imidazo[4,5-c]quinolin-4-ami...)
Affinity DataEC50:  1.21E+4nMAssay Description:Agonist activity at human TLR7 transfected in HEK cells assessed as NFkappaB induction after 24 hrs by specific secreted alkaline phosphatase gene as...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403022(CHEMBL2216760)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human TLR7 transfected in HEK cells assessed as NFkappaB induction after 24 hrs by specific secreted alkaline phosphatase gene as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403023(CHEMBL2216759)
Affinity DataEC50: >2.70E+5nMAssay Description:Agonist activity at human TLR7 transfected in HEK cells assessed as NFkappaB induction after 24 hrs by specific secreted alkaline phosphatase gene as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50320082(1-(4-Amino-2-butyl-1H-imidazo-[4,5-c]quinolin-1-yl...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human TLR7 transfected in HEK cells assessed as NFkappaB induction after 24 hrs by specific secreted alkaline phosphatase gene as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403024(CHEMBL195276)
Affinity DataEC50:  9.50E+4nMAssay Description:Agonist activity at human TLR7 transfected in HEK cells assessed as NFkappaB induction after 24 hrs by specific secreted alkaline phosphatase gene as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50241029(1-[4-amino-2-(ethoxymethyl)-1H-imidazo[4,5-c]quino...)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at human TLR7 transfected in HEK cells assessed as NFkappaB induction after 24 hrs by specific secreted alkaline phosphatase gene as...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50240849(1-(2-methylpropyl)-1H-imidazo[4,5-c]quinolin-4-ami...)
Affinity DataEC50: >2.70E+5nMAssay Description:Agonist activity at human TLR8 transfected in HEK cells assessed as NFkappaB induction after 24 hrs by specific secreted alkaline phosphatase gene as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed