Compile Data Set for Download or QSAR
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Found 16 Enz. Inhib. hit(s) with all data for entry = 50040128
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389547(CHEMBL2063984)
Affinity DataIC50:  3.47nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389547(CHEMBL2063984)
Affinity DataIC50:  3.47nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)
Affinity DataIC50:  5.62nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)
Affinity DataIC50:  6nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389544(CHEMBL2063983)
Affinity DataIC50:  24.0nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389544(CHEMBL2063983)
Affinity DataIC50:  24nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389541(CHEMBL2063979)
Affinity DataIC50:  30nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389541(CHEMBL2063979)
Affinity DataIC50:  30.2nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389542(CHEMBL2063981)
Affinity DataIC50:  117nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389542(CHEMBL2063981)
Affinity DataIC50:  117nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389545(CHEMBL2063985)
Affinity DataIC50:  245nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389545(CHEMBL2063985)
Affinity DataIC50:  245nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389543(CHEMBL2063982)
Affinity DataIC50:  446nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389543(CHEMBL2063982)
Affinity DataIC50:  447nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389546(CHEMBL2063980)
Affinity DataIC50:  631nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389546(CHEMBL2063980)
Affinity DataIC50:  634nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed