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Found 21 Enz. Inhib. hit(s) with all data for entry = 50040445
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50085041(2-(4-(3-(4-acetyl-3-hydroxy-2-propylphenoxy)propox...)
Affinity DataEC50:  650nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394344(CHEMBL2159607)
Affinity DataEC50:  3.01E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394342(CHEMBL458899)
Affinity DataEC50:  1.56E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394343(CHEMBL516827)
Affinity DataEC50:  2.93E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394345(CHEMBL2159606)
Affinity DataEC50:  1.31E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394346(CHEMBL2159605)
Affinity DataEC50:  1.10E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50085045(5-((4-((6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydro-...)
Affinity DataEC50:  720nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394341(CHEMBL465800)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394342(CHEMBL458899)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394343(CHEMBL516827)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394344(CHEMBL2159607)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394345(CHEMBL2159606)
Affinity DataEC50:  3.31E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394346(CHEMBL2159605)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50371235(CIPROFIBRATE)
Affinity DataEC50:  900nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394341(CHEMBL465800)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394342(CHEMBL458899)
Affinity DataEC50:  4.29E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394343(CHEMBL516827)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394344(CHEMBL2159607)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394345(CHEMBL2159606)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394346(CHEMBL2159605)
Affinity DataEC50:  4.71E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394341(CHEMBL465800)
Affinity DataEC50:  2.31E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed