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Found 36 Enz. Inhib. hit(s) with all data for entry = 50042493
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50315213(2-(difluoromethyl)-1-(4,6-dimorpholin-4-yl-1,3,5-t...)
Affinity DataIC50:  3nMAssay Description:Inhibition of PI3Kdelta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50315213(2-(difluoromethyl)-1-(4,6-dimorpholin-4-yl-1,3,5-t...)
Affinity DataIC50:  6nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50315213(2-(difluoromethyl)-1-(4,6-dimorpholin-4-yl-1,3,5-t...)
Affinity DataIC50:  6nMAssay Description:Inhibition of PI3Kalpha (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50315213(2-(difluoromethyl)-1-(4,6-dimorpholin-4-yl-1,3,5-t...)
Affinity DataIC50:  38nMAssay Description:Inhibition of PI3Kgamma (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426814(CHEMBL2323114)
Affinity DataIC50:  110nMAssay Description:Inhibition of PI3Kdelta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426815(CHEMBL2323117)
Affinity DataIC50:  128nMAssay Description:Inhibition of PI3Kdelta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50355706(CHEMBL1910989)
Affinity DataIC50:  187nMAssay Description:Inhibition of PI3Kdelta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426814(CHEMBL2323114)
Affinity DataIC50:  214nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50355706(CHEMBL1910989)
Affinity DataIC50:  290nMAssay Description:Inhibition of PI3Kalpha (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426814(CHEMBL2323114)
Affinity DataIC50:  375nMAssay Description:Inhibition of PI3Kalpha (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426815(CHEMBL2323117)
Affinity DataIC50:  419nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426817(CHEMBL2323119)
Affinity DataIC50:  423nMAssay Description:Inhibition of PI3Kdelta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426815(CHEMBL2323117)
Affinity DataIC50:  431nMAssay Description:Inhibition of PI3Kalpha (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426819(CHEMBL2323116)
Affinity DataIC50:  458nMAssay Description:Inhibition of PI3Kdelta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50355706(CHEMBL1910989)
Affinity DataIC50:  523nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426817(CHEMBL2323119)
Affinity DataIC50:  726nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426819(CHEMBL2323116)
Affinity DataIC50:  823nMAssay Description:Inhibition of PI3Kalpha (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426816(CHEMBL2323113)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426817(CHEMBL2323119)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426818(CHEMBL2323118)
Affinity DataIC50:  1.12E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426819(CHEMBL2323116)
Affinity DataIC50:  1.79E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50355706(CHEMBL1910989)
Affinity DataIC50:  1.86E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426815(CHEMBL2323117)
Affinity DataIC50:  2.53E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426820(CHEMBL2323115)
Affinity DataIC50:  2.77E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426816(CHEMBL2323113)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426820(CHEMBL2323115)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426818(CHEMBL2323118)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426816(CHEMBL2323113)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426820(CHEMBL2323115)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426818(CHEMBL2323118)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PI3Kalpha (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426817(CHEMBL2323119)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426818(CHEMBL2323118)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426814(CHEMBL2323114)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426820(CHEMBL2323115)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426816(CHEMBL2323113)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426819(CHEMBL2323116)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) expressed in SF21 cells using phosphatidylinositol as substrate after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed