Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for entry = 50042391
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50315537(CHEMBL1089316 | chaetocin)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50425308(CHEMBL2311579)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50425305(CHEMBL2315521)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50425304(CHEMBL2315522)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50396029(CHEMBL1222849)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50315537(CHEMBL1089316 | chaetocin)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50425311(CHEMBL2315526)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50425306(CHEMBL2315520)
Affinity DataIC50:  1.31E+4nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50425307(CHEMBL2315523)
Affinity DataIC50:  2.35E+4nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50425310(CHEMBL2315525)
Affinity DataIC50:  2.71E+4nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50396028(CHEMBL1222848)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50396028(CHEMBL1222848)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50425312(CHEMBL2315527)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50425309(CHEMBL2315524)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed