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Found 10 Enz. Inhib. hit(s) with all data for entry = 8405
TargetReplicase polyprotein 1a(Human SARS coronavirus (SARS-CoV))
Gyeongsang National University

LigandPNGBDBM246524(Psoralidin (5))
Affinity DataKi:  1.70E+3nM IC50:  4.20E+3nMpH: 8.0Assay Description:Reactions were performed in a total volume of 200 mL, which contained thefollowing components: 20mM Tris-buffer, pH 8.0, 10mM DTT, 30 mM Z-RLRGG-AMC,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1a/Z-RLRGG-AMC(Human SARS coronavirus (SARS-CoV))
Gyeongsang National University

LigandPNGBDBM246524(Psoralidin (5))
Affinity DataKi:  4.20E+3nMpH: 8.0Assay Description:Reactions were performed in a total volume of 200 mL, which contained thefollowing components: 20mM Tris-buffer, pH 8.0, 10mM DTT, 30 mM Z-RLRGG-AMC,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1a(Human SARS coronavirus (SARS-CoV))
Gyeongsang National University

LigandPNGBDBM246523(4'-O-methylbavachalcone (4))
Affinity DataKi:  4.60E+3nM IC50:  1.01E+4nMpH: 8.0Assay Description:Reactions were performed in a total volume of 200 mL, which contained thefollowing components: 20mM Tris-buffer, pH 8.0, 10mM DTT, 30 mM Z-RLRGG-AMC,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1a(Human SARS coronavirus (SARS-CoV))
Gyeongsang National University

LigandPNGBDBM50441633(4-Hydroxyisocordoin | ISOBAVACHALCONE | Isobacacha...)
Affinity DataKi:  4.90E+3nM IC50:  7.30E+3nMpH: 8.0Assay Description:Reactions were performed in a total volume of 200 mL, which contained thefollowing components: 20mM Tris-buffer, pH 8.0, 10mM DTT, 30 mM Z-RLRGG-AMC,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1a/Z-RLRGG-AMC(Human SARS coronavirus (SARS-CoV))
Gyeongsang National University

LigandPNGBDBM50441633(4-Hydroxyisocordoin | ISOBAVACHALCONE | Isobacacha...)
Affinity DataKi:  9.10E+3nMpH: 8.0Assay Description:Reactions were performed in a total volume of 200 mL, which contained thefollowing components: 20mM Tris-buffer, pH 8.0, 10mM DTT, 30 mM Z-RLRGG-AMC,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1a(Human SARS coronavirus (SARS-CoV))
Gyeongsang National University

LigandPNGBDBM246522(Neobavaisoflavone (2))
Affinity DataKi:  9.40E+3nM IC50:  1.83E+4nMpH: 8.0Assay Description:Reactions were performed in a total volume of 200 mL, which contained thefollowing components: 20mM Tris-buffer, pH 8.0, 10mM DTT, 30 mM Z-RLRGG-AMC,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1a(Human SARS coronavirus (SARS-CoV))
Gyeongsang National University

LigandPNGBDBM246525(Corylifol A (6))
Affinity DataKi:  1.14E+4nM IC50:  3.23E+4nMpH: 8.0Assay Description:Reactions were performed in a total volume of 200 mL, which contained thefollowing components: 20mM Tris-buffer, pH 8.0, 10mM DTT, 30 mM Z-RLRGG-AMC,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1a(Human SARS coronavirus (SARS-CoV))
Gyeongsang National University

LigandPNGBDBM246521(Bavachinin (1))
Affinity DataKi:  1.84E+4nM IC50:  3.84E+4nMpH: 8.0Assay Description:Reactions were performed in a total volume of 200 mL, which contained thefollowing components: 20mM Tris-buffer, pH 8.0, 10mM DTT, 30 mM Z-RLRGG-AMC,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1a(Human SARS coronavirus (SARS-CoV))
Gyeongsang National University

LigandPNGBDBM50331545(2H-furo[2,3-h]chromen-2-one | CHEMBL53569 | Furo[2...)
Affinity DataIC50: >1.50E+5nMpH: 8.0Assay Description:Reactions were performed in a total volume of 200 mL, which contained thefollowing components: 20mM Tris-buffer, pH 8.0, 10mM DTT, 30 mM Z-RLRGG-AMC,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1a(Human SARS coronavirus (SARS-CoV))
Gyeongsang National University

LigandPNGBDBM50331544(7H-furo[3,2-g]chromen-7-one | CHEMBL164660 | Furo[...)
Affinity DataIC50: >1.50E+5nMpH: 8.0Assay Description:Reactions were performed in a total volume of 200 mL, which contained thefollowing components: 20mM Tris-buffer, pH 8.0, 10mM DTT, 30 mM Z-RLRGG-AMC,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed