TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Brain Science Institute
Curated by ChEMBL
Brain Science Institute
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Modulation of mGluR5 (unknown origin)More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Brain Science Institute
Curated by ChEMBL
Brain Science Institute
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Antagonist activity at human mGluR5 expressed in HEK293 cells assessed as inhibition of L-glutamate-induced calcium mobilization by FDSS6000 assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Brain Science Institute
Curated by ChEMBL
Brain Science Institute
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Antagonist activity at human mGluR5 expressed in HEK293 cells assessed as inhibition of L-glutamate-induced calcium mobilization by FDSS6000 assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Brain Science Institute
Curated by ChEMBL
Brain Science Institute
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:Antagonist activity at human mGluR5 expressed in HEK293 cells assessed as inhibition of L-glutamate-induced calcium mobilization by FDSS6000 assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Brain Science Institute
Curated by ChEMBL
Brain Science Institute
Curated by ChEMBL
Affinity DataIC50: 940nMAssay Description:Antagonist activity at human mGluR5 expressed in HEK293 cells assessed as inhibition of L-glutamate-induced calcium mobilization by FDSS6000 assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Brain Science Institute
Curated by ChEMBL
Brain Science Institute
Curated by ChEMBL
Affinity DataIC50: 2.03E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Brain Science Institute
Curated by ChEMBL
Brain Science Institute
Curated by ChEMBL
Affinity DataIC50: 2.27E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Brain Science Institute
Curated by ChEMBL
Brain Science Institute
Curated by ChEMBL
Affinity DataIC50: 6.17E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Brain Science Institute
Curated by ChEMBL
Brain Science Institute
Curated by ChEMBL
Affinity DataIC50: 6.53E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair