Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 8413
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Msa University

LigandPNGBDBM246608(4-{4-[6-(4-(4-Bromophenyl)-3-cyano-2-imino)-1,2-di...)
Affinity DataIC50:  1.04E+3nMAssay Description:Protein kinase assays were performed at ambient temperature for 20-40 min (depending on the target) in a final volume of 25 μl according to the fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Msa University

LigandPNGBDBM246608(4-{4-[6-(4-(4-Bromophenyl)-3-cyano-2-imino)-1,2-di...)
Affinity DataIC50:  1.94E+3nMAssay Description:Protein kinase assays were performed at ambient temperature for 20-40 min (depending on the target) in a final volume of 25 μl according to the fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Msa University

LigandPNGBDBM246607(HER2/EGFR dual kinase inhibitor, 5d)
Affinity DataIC50:  2.09E+3nMAssay Description:Protein kinase assays were performed at ambient temperature for 20-40 min (depending on the target) in a final volume of 25 μl according to the fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Msa University

LigandPNGBDBM246609((E)-3-(4-Chlorophenyl)-1-{4-[(6,7-dimethoxyquinazo...)
Affinity DataIC50:  2.58E+3nMAssay Description:Protein kinase assays were performed at ambient temperature for 20-40 min (depending on the target) in a final volume of 25 μl according to the fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Msa University

LigandPNGBDBM246607(HER2/EGFR dual kinase inhibitor, 5d)
Affinity DataIC50:  3.98E+3nMAssay Description:Protein kinase assays were performed at ambient temperature for 20-40 min (depending on the target) in a final volume of 25 μl according to the fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Msa University

LigandPNGBDBM246609((E)-3-(4-Chlorophenyl)-1-{4-[(6,7-dimethoxyquinazo...)
Affinity DataIC50:  9.88E+4nMAssay Description:Protein kinase assays were performed at ambient temperature for 20-40 min (depending on the target) in a final volume of 25 μl according to the fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed