TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Antagonist activity at ERalpha receptor in human MCF7 cells assessed as inhibition of cell growth after 6 days by crystal violet staining methodMore data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]E2 from human recombinant ERalpha receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 8.70nMAssay Description:Displacement of [3H]E2 from human recombinant ERbeta receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Displacement of [3H]E2 from human recombinant ERbeta receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Displacement of [3H]E2 from human recombinant ERalpha receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Displacement of [3H]E2 from human recombinant ERalpha receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Displacement of [3H]E2 from human recombinant ERbeta receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Antagonist activity at ERalpha receptor in human MCF7 cells assessed as inhibition of cell growth after 6 days by crystal violet staining methodMore data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Antagonist activity at ERalpha receptor in human MCF7 cells assessed as inhibition of cell growth after 6 days by crystal violet staining methodMore data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Antagonist activity at ERalpha receptor in human MCF7 cells assessed as inhibition of cell growth after 6 days by crystal violet staining methodMore data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Displacement of [3H]E2 from human recombinant ERalpha receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Antagonist activity at ERalpha receptor in human MCF7 cells assessed as inhibition of cell growth after 6 days by crystal violet staining methodMore data for this Ligand-Target Pair
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 112nMAssay Description:Displacement of [3H]E2 from human recombinant ERbeta receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 116nMAssay Description:Displacement of [3H]E2 from human recombinant ERalpha receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 121nMAssay Description:Displacement of [3H]E2 from human recombinant ERbeta receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Displacement of [3H]E2 from human recombinant ERalpha receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 151nMAssay Description:Displacement of [3H]E2 from human recombinant ERbeta receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 176nMAssay Description:Displacement of [3H]E2 from human recombinant ERalpha receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 185nMAssay Description:Displacement of [3H]E2 from human recombinant ERbeta receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Antagonist activity at ERalpha receptor in human MCF7 cells assessed as inhibition of cell growth after 6 days by crystal violet staining methodMore data for this Ligand-Target Pair
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 331nMAssay Description:Displacement of [3H]E2 from human recombinant ERbeta receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 436nMAssay Description:Displacement of [3H]E2 from human recombinant ERbeta receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 482nMAssay Description:Displacement of [3H]E2 from human recombinant ERalpha receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 566nMAssay Description:Displacement of [3H]E2 from human recombinant ERbeta receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 567nMAssay Description:Displacement of [3H]E2 from human recombinant ERalpha receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
University Of Kansas Medical Center
Curated by ChEMBL
University Of Kansas Medical Center
Curated by ChEMBL
Affinity DataIC50: 638nMAssay Description:Displacement of [3H]E2 from human recombinant ERalpha receptor after overnight incubation by liquid scintillation counting analysisMore data for this Ligand-Target Pair