Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for entry = 50005342
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50491257(CHEMBL2381384)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of amyloid beta ((1 to 42) (unknown origin) oligomer assembly after 30 mins by biotinyl-streptavidin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50491252(CHEMBL2381401)
Affinity DataIC50:  1.76E+3nMAssay Description:Inhibition of AChE (unknown origin) by Ellman methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of AChE (unknown origin) by Ellman methodMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50491257(CHEMBL2381384)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) oligomer dissociation after 16 to 18 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50491254(CHEMBL2381385)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) oligomer dissociation after 16 to 18 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50491253(CHEMBL2381403)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) oligomer dissociation after 16 to 18 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50491256(CHEMBL2381400)
Affinity DataIC50:  8.27E+3nMAssay Description:Inhibition of BuChE (unknown origin) by Ellman methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of BuChE (unknown origin) by Ellman methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50491258(CHEMBL2381402)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of amyloid beta ((1 to 42) (unknown origin) oligomer assembly after 30 mins by biotinyl-streptavidin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50491253(CHEMBL2381403)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of amyloid beta ((1 to 42) (unknown origin) oligomer assembly after 30 mins by biotinyl-streptavidin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50491258(CHEMBL2381402)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) oligomer dissociation after 16 to 18 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50491254(CHEMBL2381385)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of amyloid beta ((1 to 42) (unknown origin) oligomer assembly after 30 mins by biotinyl-streptavidin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50491255(CHEMBL2381386)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of amyloid beta ((1 to 42) (unknown origin) oligomer assembly after 30 mins by biotinyl-streptavidin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University Of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50491252(CHEMBL2381401)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of amyloid beta ((1 to 42) (unknown origin) oligomer assembly after 30 mins by biotinyl-streptavidin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed