Found 80 Enz. Inhib. hit(s) with all data for entry = 50005437 TargetAdenosine receptor A1(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 0.580nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 6.70nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 9.40nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 75nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 128nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 177nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 179nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 193nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 201nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 276nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 327nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 406nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 536nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 552nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 562nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 567nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 676nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 688nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 746nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 801nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 816nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 841nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 918nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 951nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 1.38E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 1.87E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 2.01E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 2.04E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 2.47E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 2.64E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 3.63E+3nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 3.93E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 4.87E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 5.95E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 7.24E+3nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 8.00E+3nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 8.78E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 9.11E+3nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
