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Found 36 Enz. Inhib. hit(s) with all data for entry = 50043342
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM11695((2S)-1-{2-[(3-hydroxyadamantan-1-yl)amino]acetyl}p...)
Affinity DataIC50:  66nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439572(CHEMBL2418633)
Affinity DataIC50:  240nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439572(CHEMBL2418633)
Affinity DataIC50:  260nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439585(CHEMBL2418637)
Affinity DataIC50:  280nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439579(CHEMBL2418627)
Affinity DataIC50:  280nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439575(CHEMBL2418630)
Affinity DataIC50:  300nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439575(CHEMBL2418630)
Affinity DataIC50:  310nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439578(CHEMBL2417563)
Affinity DataIC50:  320nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439582(CHEMBL2418624)
Affinity DataIC50:  330nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439574(CHEMBL2418631)
Affinity DataIC50:  330nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439577(CHEMBL2418628)
Affinity DataIC50:  340nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439577(CHEMBL2418628)
Affinity DataIC50:  340nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439582(CHEMBL2418624)
Affinity DataIC50:  340nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439578(CHEMBL2417563)
Affinity DataIC50:  350nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439581(CHEMBL2418625)
Affinity DataIC50:  360nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439579(CHEMBL2418627)
Affinity DataIC50:  390nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439581(CHEMBL2418625)
Affinity DataIC50:  430nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439580(CHEMBL2418626)
Affinity DataIC50:  440nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439573(CHEMBL2418632)
Affinity DataIC50:  440nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439580(CHEMBL2418626)
Affinity DataIC50:  440nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439574(CHEMBL2418631)
Affinity DataIC50:  450nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439583(CHEMBL2418639)
Affinity DataIC50:  450nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439571(CHEMBL2418634)
Affinity DataIC50:  470nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439583(CHEMBL2418639)
Affinity DataIC50:  510nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439576(CHEMBL2418629)
Affinity DataIC50:  550nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439571(CHEMBL2418634)
Affinity DataIC50:  600nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439585(CHEMBL2418637)
Affinity DataIC50:  620nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439586(CHEMBL2418636)
Affinity DataIC50:  630nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439586(CHEMBL2418636)
Affinity DataIC50:  680nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439573(CHEMBL2418632)
Affinity DataIC50:  690nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM11695((2S)-1-{2-[(3-hydroxyadamantan-1-yl)amino]acetyl}p...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439584(CHEMBL2418638)
Affinity DataIC50:  1.13E+3nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439576(CHEMBL2418629)
Affinity DataIC50:  1.21E+3nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50439584(CHEMBL2418638)
Affinity DataIC50:  1.61E+3nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)
Affinity DataIC50:  1.15E+5nMAssay Description:Inhibition of human purified His-tagged DPP-8 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)
Affinity DataIC50:  1.30E+5nMAssay Description:Inhibition of human purified His-tagged DPP-9 assessed as cleavage of substrate using Gly-Pro-AMC chromogenic substrate after 60 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed