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Found 10 Enz. Inhib. hit(s) with all data for entry = 50043391
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50440393(CHEMBL2425487)
Affinity DataIC50:  24nMAssay Description:Inhibition of recombinant CDK5/p25 (unknown origin) expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50077360(3,10-Dihydroxy-13-(3-hydroxy-4-methoxy-phenyl)-2,1...)
Affinity DataIC50:  25nMAssay Description:Inhibition of recombinant CDK5/p25 (unknown origin) expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50077360(3,10-Dihydroxy-13-(3-hydroxy-4-methoxy-phenyl)-2,1...)
Affinity DataIC50:  35nMAssay Description:Inhibition of human recombinant DYRK1A expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50077360(3,10-Dihydroxy-13-(3-hydroxy-4-methoxy-phenyl)-2,1...)
Affinity DataIC50:  55nMAssay Description:Inhibition of PIM1 (unknown origin) expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK3(Mus musculus)
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50440393(CHEMBL2425487)
Affinity DataIC50:  150nMAssay Description:Inhibition of mouse recombinant CLK3 expressed in Escherichia coli using RS peptide and [gamma-33P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50440393(CHEMBL2425487)
Affinity DataIC50:  220nMAssay Description:Inhibition of PIM1 (unknown origin) expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50440393(CHEMBL2425487)
Affinity DataIC50:  220nMAssay Description:Inhibition of PIM1 (unknown origin) expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50440393(CHEMBL2425487)
Affinity DataIC50:  440nMAssay Description:Inhibition of human recombinant DYRK1A expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50440393(CHEMBL2425487)
Affinity DataIC50:  440nMAssay Description:Inhibition of human recombinant DYRK1A expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK3(Mus musculus)
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50440393(CHEMBL2425487)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mouse recombinant CLK3 expressed in Escherichia coli using RS peptide and [gamma-33P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed