Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50043393
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Leopold-Franzens-Universit£T

Curated by ChEMBL
LigandPNGBDBM50440407(CHEMBL2425589)
Affinity DataIC50:  700nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells assessed as [1,2-3H]-cortisone reduction to [1,2,6,7-3H]-cortisol after 10 mins in presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Leopold-Franzens-Universit£T

Curated by ChEMBL
LigandPNGBDBM50440405(CHEMBL2425591)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells assessed as [1,2-3H]-cortisone reduction to [1,2,6,7-3H]-cortisol after 10 mins in presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Leopold-Franzens-Universit£T

Curated by ChEMBL
LigandPNGBDBM50440406(CHEMBL2425590)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells assessed as [1,2-3H]-cortisone reduction to [1,2,6,7-3H]-cortisol after 10 mins in presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Leopold-Franzens-Universit£T

Curated by ChEMBL
LigandPNGBDBM50440408(CHEMBL2425588)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells assessed as [1,2-3H]-cortisone reduction to [1,2,6,7-3H]-cortisol after 10 mins in presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Leopold-Franzens-Universit£T

Curated by ChEMBL
LigandPNGBDBM50440404(CHEMBL2425592)
Affinity DataIC50:  1.85E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells assessed as [1,2-3H]-cortisone reduction to [1,2,6,7-3H]-cortisol after 10 mins in presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Leopold-Franzens-Universit£T

Curated by ChEMBL
LigandPNGBDBM50440403(CHEMBL2425593)
Affinity DataIC50:  2.72E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells assessed as [1,2-3H]-cortisone reduction to [1,2,6,7-3H]-cortisol after 10 mins in presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed