Compile Data Set for Download or QSAR
maximum 50k data
Found 38 Enz. Inhib. hit(s) with all data for entry = 6210
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115198(10‐(4‐bromobenzenesulfonyl)‐N...)
Affinity DataIC50:  2.80E+3nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115182(N‐(4‐ethoxyphenyl)‐8‐metho...)
Affinity DataIC50:  3.30E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115184(8‐methoxy‐N‐(4‐methoxyphen...)
Affinity DataIC50:  3.50E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115190(2‐(2‐{[(5E)‐2‐imino‐...)
Affinity DataIC50:  3.70E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115185(8‐methoxy‐N‐[3‐(methylsulf...)
Affinity DataIC50:  3.80E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM50322180(3-(2,5-dimethylphenylsulfonyl)-N-isopropylthieno[2...)
Affinity DataIC50:  3.80E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115194(4‐(4,5‐dihydro‐1,3‐thiazol...)
Affinity DataIC50:  4.20E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115191((5E)‐5‐[(2‐hydroxy‐3‐...)
Affinity DataIC50:  4.60E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115190(2‐(2‐{[(5E)‐2‐imino‐...)
Affinity DataIC50:  4.80E+3nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115183(8‐hydroxy‐N‐[(3‐methoxyphe...)
Affinity DataIC50:  5.30E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115193((5E)‐5‐[(4‐hydroxy‐3‐...)
Affinity DataIC50:  6.20E+3nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115184(8‐methoxy‐N‐(4‐methoxyphen...)
Affinity DataIC50:  6.20E+3nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115191((5E)‐5‐[(2‐hydroxy‐3‐...)
Affinity DataIC50:  6.30E+3nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115192((5E)‐5‐[(2,3‐dimethoxyphenyl)met...)
Affinity DataIC50:  7.00E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM50322180(3-(2,5-dimethylphenylsulfonyl)-N-isopropylthieno[2...)
Affinity DataIC50:  1.50E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115182(N‐(4‐ethoxyphenyl)‐8‐metho...)
Affinity DataIC50:  1.60E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115187(N‐(3‐chloro‐4‐methoxypheny...)
Affinity DataIC50:  1.90E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115185(8‐methoxy‐N‐[3‐(methylsulf...)
Affinity DataIC50:  2.00E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115188(N‐(3‐chloro‐4‐methylphenyl...)
Affinity DataIC50:  2.40E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115186(N‐(4‐ethoxyphenyl)‐8‐metho...)
Affinity DataIC50:  2.40E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115193((5E)‐5‐[(4‐hydroxy‐3‐...)
Affinity DataIC50:  2.50E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115189(N‐(3‐fluoro‐4‐methylphenyl...)
Affinity DataIC50:  2.50E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115187(N‐(3‐chloro‐4‐methoxypheny...)
Affinity DataIC50:  2.70E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM50322183(3-(4-ethylphenylsulfonyl)-N-(3-methoxypropyl)thien...)
Affinity DataIC50:  2.80E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115186(N‐(4‐ethoxyphenyl)‐8‐metho...)
Affinity DataIC50:  3.40E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115197(10‐(benzenesulfonyl)‐N‐methyl...)
Affinity DataIC50:  3.50E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115196(2‐N‐(3‐methoxyphenyl)‐4...)
Affinity DataIC50:  4.20E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115192((5E)‐5‐[(2,3‐dimethoxyphenyl)met...)
Affinity DataIC50:  4.30E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115195(1‐N‐[bis(methylsulfanyl)‐1,3,5&#...)
Affinity DataIC50:  4.50E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115194(4‐(4,5‐dihydro‐1,3‐thiazol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115195(1‐N‐[bis(methylsulfanyl)‐1,3,5&#...)
Affinity DataIC50: >5.00E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115196(2‐N‐(3‐methoxyphenyl)‐4...)
Affinity DataIC50: >5.00E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115198(10‐(4‐bromobenzenesulfonyl)‐N...)
Affinity DataIC50: >5.00E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM50322183(3-(4-ethylphenylsulfonyl)-N-(3-methoxypropyl)thien...)
Affinity DataIC50: >5.00E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115189(N‐(3‐fluoro‐4‐methylphenyl...)
Affinity DataIC50: >5.00E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115188(N‐(3‐chloro‐4‐methylphenyl...)
Affinity DataIC50: >5.00E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115183(8‐hydroxy‐N‐[(3‐methoxyphe...)
Affinity DataIC50: >5.00E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115197(10‐(benzenesulfonyl)‐N‐methyl...)
Affinity DataIC50: >5.00E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed