Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50044310
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50035131((+)-(6R,11S)-6,11-dimethyl-3-(3-methyl-but-2-enyl)...)
Affinity DataKi:  2.60nMAssay Description:Displacement of (+)-[3H]pentazocine from Dunkin guinea pig brain sigma 1 receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50012204(CHEMBL3259962)
Affinity DataKi:  5.40nMAssay Description:Displacement of (+)-[3H]pentazocine from Dunkin guinea pig brain sigma 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50012203(CHEMBL3259961)
Affinity DataKi:  156nMAssay Description:Displacement of (+)-[3H]pentazocine from Dunkin guinea pig brain sigma 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50012205(CHEMBL3259963)
Affinity DataKi:  235nMAssay Description:Displacement of (+)-[3H]pentazocine from Dunkin guinea pig brain sigma 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50012192(CHEMBL3259960)
Affinity DataKi:  258nMAssay Description:Displacement of (+)-[3H]pentazocine from Dunkin guinea pig brain sigma 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed