Compile Data Set for Download or QSAR
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Found 9 Enz. Inhib. hit(s) with all data for entry = 50005543
TargetHistone deacetylase 4(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM187543(US9670193, 21 (R)?N-(1-(benzyl(methyl)amino)propan...)
Affinity DataIC50:  18nMAssay Description:Inhibition of recombinant human HDAC-4 (2 to 1084) expressed in baculovirus infected Sf9 cells using acetyl-Gly-Ala-Lys(E-trifluoroacetyl)-AMC as sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM187565(US9670193, 23 (R)?N-(1-(diethylamino)propan-2-yl)-...)
Affinity DataIC50:  28nMAssay Description:Inhibition of recombinant human HDAC-4 (2 to 1084) expressed in baculovirus infected Sf9 cells using acetyl-Gly-Ala-Lys(E-trifluoroacetyl)-AMC as sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM187220(US9670193, 10 N-(pyridin-3-ylmethyl)-5-(5-(trifluo...)
Affinity DataIC50:  140nMAssay Description:Inhibition of recombinant human HDAC-4 (2 to 1084) expressed in baculovirus infected Sf9 cells using acetyl-Gly-Ala-Lys(E-trifluoroacetyl)-AMC as sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM187220(US9670193, 10 N-(pyridin-3-ylmethyl)-5-(5-(trifluo...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of recombinant full length human HDAC-6 expressed in baculovirus expression system using acetyl-Gly-Ala-Lys(acetyl)-AMC as substrate after...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM187220(US9670193, 10 N-(pyridin-3-ylmethyl)-5-(5-(trifluo...)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of recombinant full length human HDAC-1 expressed in baculovirus expression system using acetyl-Gly-Ala-Lys(acetyl)-AMC as substrate after...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM187543(US9670193, 21 (R)?N-(1-(benzyl(methyl)amino)propan...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant full length human HDAC-1 expressed in baculovirus expression system using acetyl-Gly-Ala-Lys(acetyl)-AMC as substrate after...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM187543(US9670193, 21 (R)?N-(1-(benzyl(methyl)amino)propan...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant full length human HDAC-6 expressed in baculovirus expression system using acetyl-Gly-Ala-Lys(acetyl)-AMC as substrate after...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM187565(US9670193, 23 (R)?N-(1-(diethylamino)propan-2-yl)-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant full length human HDAC-6 expressed in baculovirus expression system using acetyl-Gly-Ala-Lys(acetyl)-AMC as substrate after...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM187565(US9670193, 23 (R)?N-(1-(diethylamino)propan-2-yl)-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant full length human HDAC-1 expressed in baculovirus expression system using acetyl-Gly-Ala-Lys(acetyl)-AMC as substrate after...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed