Compile Data Set for Download or QSAR
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Found 48 Enz. Inhib. hit(s) with all data for entry = 50044674
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025019(CHEMBL3337845)
Affinity DataIC50:  10nMAssay Description:Inhibition of rat CK1delta kinetic domain expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025016(CHEMBL3337849)
Affinity DataIC50:  18nMAssay Description:Inhibition of rat CK1delta by radiometric protein kinase filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025019(CHEMBL3337845)
Affinity DataIC50:  20nMAssay Description:Inhibition of rat CK1delta kinetic domain expressed in Escherichia coli using alpha casein substrate by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025019(CHEMBL3337845)
Affinity DataIC50:  20nMAssay Description:Inhibition of GST-tagged rat CK1delta expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025020(CHEMBL3337854)
Affinity DataIC50:  29nMAssay Description:Inhibition of rat CK1delta kinetic domain expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025015(CHEMBL3337846)
Affinity DataIC50:  34nMAssay Description:Inhibition of rat CK1delta by radiometric protein kinase filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025020(CHEMBL3337854)
Affinity DataIC50:  40nMAssay Description:Inhibition of GST-tagged rat CK1delta expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025015(CHEMBL3337846)
Affinity DataIC50:  70nMAssay Description:Inhibition of rat CK1delta kinetic domain expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025019(CHEMBL3337845)
Affinity DataIC50:  70nMAssay Description:Inhibition of GST-tagged rat CK1delta expressed in Escherichia coli using alpha casein substrate by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025017(CHEMBL3337855)
Affinity DataIC50:  106nMAssay Description:Inhibition of rat CK1delta by radiometric protein kinase filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025015(CHEMBL3337846)
Affinity DataIC50:  130nMAssay Description:Inhibition of GST-tagged rat CK1delta expressed in Escherichia coli using alpha casein substrate by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025024(CHEMBL3337850)
Affinity DataIC50:  130nMAssay Description:Inhibition of GST-tagged rat CK1delta expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025015(CHEMBL3337846)
Affinity DataIC50:  140nMAssay Description:Inhibition of GST-tagged rat CK1delta expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Bos taurus)
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025019(CHEMBL3337845)
Affinity DataIC50:  160nMAssay Description:Inhibition of GST-tagged bovine CK1alpha expressed in Escherichia coli using alpha casein substrate by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025015(CHEMBL3337846)
Affinity DataIC50:  160nMAssay Description:Inhibition of human recombinant CK1epsilon expressed in Escherichia coli using alpha casein substrate by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025015(CHEMBL3337846)
Affinity DataIC50:  170nMAssay Description:Inhibition of rat CK1delta kinetic domain expressed in Escherichia coli using alpha casein substrate by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025023(CHEMBL3337851)
Affinity DataIC50:  180nMAssay Description:Inhibition of rat CK1delta kinetic domain expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025016(CHEMBL3337849)
Affinity DataIC50:  180nMAssay Description:Inhibition of rat CK1delta kinetic domain expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025019(CHEMBL3337845)
Affinity DataIC50:  190nMAssay Description:Inhibition of human recombinant CK1epsilon expressed in Escherichia coli using alpha casein substrate by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025020(CHEMBL3337854)
Affinity DataIC50:  199nMAssay Description:Inhibition of human recombinant CK1epsilon expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025018(CHEMBL3337856)
Affinity DataIC50:  201nMAssay Description:Inhibition of rat CK1delta by radiometric protein kinase filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025016(CHEMBL3337849)
Affinity DataIC50:  210nMAssay Description:Inhibition of GST-tagged rat CK1delta expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025019(CHEMBL3337845)
Affinity DataIC50:  210nMAssay Description:Inhibition of human recombinant CK1epsilon expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025023(CHEMBL3337851)
Affinity DataIC50:  260nMAssay Description:Inhibition of GST-tagged rat CK1delta expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025026(CHEMBL3337847)
Affinity DataIC50:  270nMAssay Description:Inhibition of rat CK1delta kinetic domain expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025024(CHEMBL3337850)
Affinity DataIC50:  290nMAssay Description:Inhibition of rat CK1delta kinetic domain expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025022(CHEMBL3337852)
Affinity DataIC50:  300nMAssay Description:Inhibition of GST-tagged rat CK1delta expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025023(CHEMBL3337851)
Affinity DataIC50:  320nMAssay Description:Inhibition of human recombinant CK1epsilon expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025022(CHEMBL3337852)
Affinity DataIC50:  350nMAssay Description:Inhibition of rat CK1delta kinetic domain expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025024(CHEMBL3337850)
Affinity DataIC50:  420nMAssay Description:Inhibition of human recombinant CK1epsilon expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025016(CHEMBL3337849)
Affinity DataIC50:  460nMAssay Description:Inhibition of human recombinant CK1epsilon expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025021(CHEMBL3337853)
Affinity DataIC50:  520nMAssay Description:Inhibition of rat CK1delta kinetic domain expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025015(CHEMBL3337846)
Affinity DataIC50:  520nMAssay Description:Inhibition of human recombinant CK1epsilon expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025021(CHEMBL3337853)
Affinity DataIC50:  550nMAssay Description:Inhibition of GST-tagged rat CK1delta expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025026(CHEMBL3337847)
Affinity DataIC50:  560nMAssay Description:Inhibition of GST-tagged rat CK1delta expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025025(CHEMBL3337848)
Affinity DataIC50:  570nMAssay Description:Inhibition of GST-tagged rat CK1delta expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025022(CHEMBL3337852)
Affinity DataIC50:  600nMAssay Description:Inhibition of human recombinant CK1epsilon expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025021(CHEMBL3337853)
Affinity DataIC50:  620nMAssay Description:Inhibition of human recombinant CK1epsilon expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025025(CHEMBL3337848)
Affinity DataIC50:  750nMAssay Description:Inhibition of rat CK1delta kinetic domain expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform gamma-3(Homo sapiens (Human))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025015(CHEMBL3337846)
Affinity DataIC50:  800nMAssay Description:Inhibition of GST-tagged human CK1gamma3 expressed in Escherichia coli using using alpha casein substrate by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform gamma-3(Homo sapiens (Human))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025019(CHEMBL3337845)
Affinity DataIC50:  810nMAssay Description:Inhibition of GST-tagged human CK1gamma3 expressed in Escherichia coli using using alpha casein substrate by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025026(CHEMBL3337847)
Affinity DataIC50:  990nMAssay Description:Inhibition of human recombinant CK1epsilon expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Bos taurus)
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025015(CHEMBL3337846)
Affinity DataIC50:  1.36E+3nMAssay Description:Inhibition of GST-tagged bovine CK1alpha expressed in Escherichia coli using alpha casein substrate by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025025(CHEMBL3337848)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CK1epsilon expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025019(CHEMBL3337845)
Affinity DataIC50:  2.01E+4nMAssay Description:Inhibition of GST-tagged mouse CK1delta transcription variant 1 mutant expressed in Escherichia coli at 15 degC for 14 hrs using GST-p53 (1 to 64 res...More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025019(CHEMBL3337845)
Affinity DataIC50:  3.66E+4nMAssay Description:Inhibition of GST-tagged mouse CK1delta transcription variant 2 mutant expressed in Escherichia coli at 15 degC for 14 hrs using GST-p53 (1 to 64 res...More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025019(CHEMBL3337845)
Affinity DataIC50:  5.59E+4nMAssay Description:Inhibition of GST-tagged mouse CK1delta transcription variant 2 mutant expressed in Escherichia coli at 37 degC for 2 hrs using GST-p53 (1 to 64 resi...More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50025019(CHEMBL3337845)
Affinity DataIC50:  8.01E+4nMAssay Description:Inhibition of GST-tagged mouse CK1delta transcription variant 1 mutant expressed in Escherichia coli at 37 degC for 2 hrs using GST-p53 (1 to 64 resi...More data for this Ligand-Target Pair