Compile Data Set for Download or QSAR
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Found 35 Enz. Inhib. hit(s) with all data for entry = 50006165
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50340753(2-(4-(2-(4-chlorophenethylamino)pyrimidin-4-yl)pip...)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497465(CHEMBL3343995)
Affinity DataIC50:  800nMAssay Description:Antagonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Rattus norvegicus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Mus musculus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497460(CHEMBL3343988)
Affinity DataEC50:  794nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Mus musculus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50:  3.16E+4nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497461(CHEMBL3343990)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50336912(Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497460(CHEMBL3343988)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497462(CHEMBL3343987)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Rattus norvegicus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497461(CHEMBL3343990)
Affinity DataEC50:  6.31E+3nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Rattus norvegicus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50412987(CHEMBL475965)
Affinity DataEC50: <2.00E+3nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Rattus norvegicus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497462(CHEMBL3343987)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Rattus norvegicus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497463(CHEMBL3343991)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Rattus norvegicus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497464(CHEMBL3343993)
Affinity DataEC50:  5.01E+4nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Mus musculus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497461(CHEMBL3343990)
Affinity DataEC50:  501nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Mus musculus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497462(CHEMBL3343987)
Affinity DataEC50:  7.94E+3nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Mus musculus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497463(CHEMBL3343991)
Affinity DataEC50:  501nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Mus musculus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50:  3.16E+4nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Mus musculus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497458(CHEMBL3343994)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50412987(CHEMBL475965)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Rattus norvegicus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM224021(BAM8-22 | VGRPEWWMDYQKRYG)
Affinity DataEC50:  316nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497464(CHEMBL3343993)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Rattus norvegicus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497458(CHEMBL3343994)
Affinity DataEC50:  631nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Rattus norvegicus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497460(CHEMBL3343988)
Affinity DataEC50:  3.98E+3nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Mus musculus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50412987(CHEMBL475965)
Affinity DataEC50: <2.00E+3nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Mus musculus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497464(CHEMBL3343993)
Affinity DataEC50:  1.58E+4nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Mus musculus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM224021(BAM8-22 | VGRPEWWMDYQKRYG)
Affinity DataEC50:  251nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497463(CHEMBL3343991)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Rattus norvegicus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Rattus norvegicus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50336912(Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...)
Affinity DataEC50:  6.31E+3nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497458(CHEMBL3343994)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Mus musculus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50336912(Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...)
Affinity DataEC50:  316nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM224021(BAM8-22 | VGRPEWWMDYQKRYG)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed