Affinity DataKi: 0.0300nMAssay Description:Binding affinity to recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Binding affinity to recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity to recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity to recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity to recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Binding affinity to recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Binding affinity to recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.30nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.60nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.20nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 103nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 384nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.36E+3nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4.80nMAssay Description:Antagonist activity at recombinant human H3 receptor expressed on CHO-K1 cells assessed as cAMP level by luciferase gene reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Antagonist activity at recombinant human H3 receptor expressed on CHO-K1 cells assessed as cAMP level by luciferase gene reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 274nMAssay Description:Antagonist activity at recombinant human H3 receptor expressed on CHO-K1 cells assessed as cAMP level by luciferase gene reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 324nMAssay Description:Antagonist activity at recombinant human H3 receptor expressed on CHO-K1 cells assessed as cAMP level by luciferase gene reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 459nMAssay Description:Antagonist activity at recombinant human H3 receptor expressed on CHO-K1 cells assessed as cAMP level by luciferase gene reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human CYP2D6 after 12 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human CYP3A4 after 2 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >4.50E+4nMAssay Description:Inhibition of human CYP3A4 after 2 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >4.50E+4nMAssay Description:Inhibition of human CYP2D6 after 12 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair