Compile Data Set for Download or QSAR
maximum 50k data
Found 26 Enz. Inhib. hit(s) with all data for entry = 50010186
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50529668(Enobosarm | Gtx-024 | MK-2866 | Ostarine | US10806...)
Affinity DataIC50:  36nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535824(CHEMBL4575144)
Affinity DataIC50:  49nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535836(CHEMBL4558169)
Affinity DataIC50:  59nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535830(CHEMBL4523011)
Affinity DataIC50:  72nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535839(CHEMBL4577418)
Affinity DataIC50:  80nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535835(CHEMBL4547536)
Affinity DataIC50:  111nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535841(CHEMBL4529395)
Affinity DataIC50:  123nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535837(CHEMBL4482919)
Affinity DataIC50:  183nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535829(CHEMBL4529026)
Affinity DataIC50:  198nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535825(CHEMBL4572299)
Affinity DataIC50:  245nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535834(CHEMBL4532289)
Affinity DataIC50:  265nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535826(CHEMBL4581453)
Affinity DataIC50:  280nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535827(CHEMBL4580745)
Affinity DataIC50:  332nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50425732(ENZALUTAMIDE | US10053433, FC 4.129 | US10806720, ...)
Affinity DataIC50:  361nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535840(CHEMBL4533483)
Affinity DataIC50:  402nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535843(CHEMBL4589154)
Affinity DataIC50:  407nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535823(CHEMBL4483683)
Affinity DataIC50:  425nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM18678((2R)-N-[4-cyano-3-(trifluoromethyl)phenyl]-3-[(4-f...)
Affinity DataIC50:  490nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535842(CHEMBL4572778)
Affinity DataIC50:  625nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535828(CHEMBL4519421)
Affinity DataIC50:  625nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535831(CHEMBL4516292)
Affinity DataIC50:  736nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535832(CHEMBL4585541)
Affinity DataIC50:  775nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535833(CHEMBL4521612)
Affinity DataIC50:  777nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535844(CHEMBL4537113)
Affinity DataIC50:  811nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535845(CHEMBL4549022)
Affinity DataIC50:  1.07E+3nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
School Of Pharmacy And Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535838(CHEMBL4556247)
Affinity DataIC50:  2.17E+3nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed