Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 7414
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  54nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193713(Pyrimidin-4-one-1,2,3-triazole conjugate, 3n)
Affinity DataIC50:  82nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193706(Pyrimidin-4-one-1,2,3-triazole conjugate, 3g)
Affinity DataIC50:  94nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193709(Pyrimidin-4-one-1,2,3-triazole conjugate, 3j)
Affinity DataIC50:  122nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193717(Pyrimidin-4-one-1,2,3-triazole conjugate, 3r)
Affinity DataIC50:  153nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193701(Pyrimidin-4-one-1,2,3-triazole conjugate, 3b)
Affinity DataIC50:  200nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193703(Pyrimidin-4-one-1,2,3-triazole conjugate, 3d)
Affinity DataIC50:  302nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193702(Pyrimidin-4-one-1,2,3-triazole conjugate, 3c)
Affinity DataIC50:  437nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193710(Pyrimidin-4-one-1,2,3-triazole conjugate, 3k)
Affinity DataIC50:  502nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193712(Pyrimidin-4-one-1,2,3-triazole conjugate, 3m)
Affinity DataIC50:  577nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193716(Pyrimidin-4-one-1,2,3-triazole conjugate, 3q)
Affinity DataIC50:  587nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193700(Pyrimidin-4-one-1,2,3-triazole conjugate, 3a)
Affinity DataIC50:  744nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193704(Pyrimidin-4-one-1,2,3-triazole conjugate, 3e)
Affinity DataIC50:  916nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193714(Pyrimidin-4-one-1,2,3-triazole conjugate, 3o)
Affinity DataIC50:  1.14E+3nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193708(Pyrimidin-4-one-1,2,3-triazole conjugate, 3i)
Affinity DataIC50:  1.31E+3nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193705(Pyrimidin-4-one-1,2,3-triazole conjugate, 3f)
Affinity DataIC50:  1.34E+3nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193707(Pyrimidin-4-one-1,2,3-triazole conjugate, 3h)
Affinity DataIC50:  1.44E+3nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193715(Pyrimidin-4-one-1,2,3-triazole conjugate, 3p)
Affinity DataIC50:  1.56E+3nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

LigandPNGBDBM193711(Pyrimidin-4-one-1,2,3-triazole conjugate, 3l)
Affinity DataIC50:  1.74E+3nMAssay Description:In a typical assay, 10 無 of test compound of different concentrations (dissolved in dimethyl sulfoxide [DMSO] and diluted with assay buffer) and 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed