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Found 29 Enz. Inhib. hit(s) with all data for entry = 50048264
TargetCholinesterase(Equus caballus (Horse))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210854(CHEMBL3960040)
Affinity DataKi:  0.700nMAssay Description:Competitive inhibition of horse serum BChE in presence of varying levels of butyrylthiocholine iodide substrate by Lineweaver-burk plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210854(CHEMBL3960040)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of horse serum BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210854(CHEMBL3960040)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of human BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210852(CHEMBL3971112)
Affinity DataIC50:  13nMAssay Description:Inhibition of human BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210852(CHEMBL3971112)
Affinity DataIC50:  24nMAssay Description:Inhibition of horse serum BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210848(CHEMBL3907854)
Affinity DataIC50:  28nMAssay Description:Inhibition of horse serum BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210847(CHEMBL3889911)
Affinity DataIC50:  65nMAssay Description:Inhibition of horse serum BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210842(CHEMBL3919289)
Affinity DataIC50:  230nMAssay Description:Inhibition of horse serum BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  560nMAssay Description:Inhibition of electric eel AChE pretreated for 20 mins followed by acetylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210768(CHEMBL3914751)
Affinity DataIC50:  1.14E+3nMAssay Description:Inhibition of horse serum BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210849(CHEMBL3962431)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of horse serum BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210842(CHEMBL3919289)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210851(CHEMBL3962358)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of horse serum BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210851(CHEMBL3962358)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of electric eel AChE pretreated for 20 mins followed by acetylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210842(CHEMBL3919289)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human AChE pretreated for 20 mins followed by acetylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210855(CHEMBL3935090)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibition of electric eel AChE pretreated for 20 mins followed by acetylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210844(CHEMBL3937926)
Affinity DataIC50:  1.07E+4nMAssay Description:Inhibition of horse serum BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  1.19E+4nMAssay Description:Inhibition of horse serum BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210855(CHEMBL3935090)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of horse serum BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210852(CHEMBL3971112)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of human AChE pretreated for 20 mins followed by acetylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210843(CHEMBL3971444)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of horse serum BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210852(CHEMBL3971112)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of electric eel AChE pretreated for 20 mins followed by acetylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210846(CHEMBL3910836)
Affinity DataIC50:  2.23E+4nMAssay Description:Inhibition of horse serum BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210853(CHEMBL3900327)
Affinity DataIC50:  2.57E+4nMAssay Description:Inhibition of horse serum BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210845(CHEMBL3892498)
Affinity DataIC50:  4.48E+4nMAssay Description:Inhibition of electric eel AChE pretreated for 20 mins followed by acetylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210853(CHEMBL3900327)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of electric eel AChE pretreated for 20 mins followed by acetylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210850(CHEMBL3979295)
Affinity DataIC50:  6.82E+4nMAssay Description:Inhibition of horse serum BChE pretreated for 20 mins followed by butyrylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210846(CHEMBL3910836)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of electric eel AChE pretreated for 20 mins followed by acetylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bari&Quot;A. Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50210843(CHEMBL3971444)
Affinity DataIC50:  1.10E+5nMAssay Description:Inhibition of electric eel AChE pretreated for 20 mins followed by acetylthiocholine iodide substrate addition measured for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed