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Found 66 Enz. Inhib. hit(s) with all data for entry = 50049277
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237925(CHEMBL4103223)
Affinity DataIC50:  580nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237961(CHEMBL4060753)
Affinity DataIC50:  850nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237964(CHEMBL4090465)
Affinity DataIC50:  920nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237931(CHEMBL4095459)
Affinity DataIC50:  920nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237942(CHEMBL4078955)
Affinity DataIC50:  1.07E+3nMAssay Description:Displacement of [3H]dexamethasone from human Glucocorticoid receptor (GR); Value ranges from 44-53 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237915(CHEMBL4069435)
Affinity DataIC50:  1.11E+3nMAssay Description:Inhibition of human IAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237939(CHEMBL4077330)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237962(CHEMBL4079164)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237920(CHEMBL4087225)
Affinity DataIC50:  1.33E+3nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237915(CHEMBL4069435)
Affinity DataIC50:  1.33E+3nMAssay Description:Effect on functional cellular GR-antagonism (GRAF) in human Glucocorticoid receptor (GR) expressing cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237946(CHEMBL4105082)
Affinity DataIC50:  1.33E+3nMAssay Description:Displacement of [3H]dexamethasone from human Glucocorticoid receptor (GR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237965(CHEMBL4068298)
Affinity DataIC50:  1.42E+3nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237928(CHEMBL4084312)
Affinity DataIC50:  1.64E+3nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237916(CHEMBL4094534)
Affinity DataIC50:  1.83E+3nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237923(CHEMBL4075025)
Affinity DataIC50:  1.94E+3nMAssay Description:Effect on human Glucocorticoid receptor (GR) in a whole cell assay to measure functional cellular GR-antagonism (GRAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237963(CHEMBL4098180)
Affinity DataIC50:  1.99E+3nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237922(CHEMBL4103420)
Affinity DataIC50:  2.13E+3nMAssay Description:Displacement of [3H]dexamethasone from human Glucocorticoid receptor (GR); Value ranges from 3-4 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237937(CHEMBL1372043)
Affinity DataIC50:  2.16E+3nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237926(CHEMBL4080152)
Affinity DataIC50:  2.26E+3nMAssay Description:Inhibition of human IAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237918(CHEMBL4093867)
Affinity DataIC50:  2.31E+3nMAssay Description:Effect on human Glucocorticoid receptor (GR) in a whole cell assay to measure functional cellular GR-antagonism (GRAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237913(CHEMBL4091160)
Affinity DataIC50:  2.42E+3nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237926(CHEMBL4080152)
Affinity DataIC50:  2.47E+3nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237941(CHEMBL4073985)
Affinity DataIC50:  2.51E+3nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237945(CHEMBL4070218)
Affinity DataIC50:  2.52E+3nMAssay Description:Agonistic activity measures the ability to induce alkaline phosphatase in T47D human breast cancer cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237966(CHEMBL4078377)
Affinity DataIC50:  2.54E+3nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237924(CHEMBL4102277)
Affinity DataIC50:  2.56E+3nMAssay Description:Effect on human Glucocorticoid receptor (GR) in a whole cell assay to measure functional cellular GR-antagonism (GRAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237967(CHEMBL4073185)
Affinity DataIC50:  2.59E+3nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237918(CHEMBL4093867)
Affinity DataIC50:  2.72E+3nMAssay Description:Inhibition of human IAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237964(CHEMBL4090465)
Affinity DataIC50:  2.81E+3nMAssay Description:Inhibition of human IAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237923(CHEMBL4075025)
Affinity DataIC50:  2.87E+3nMAssay Description:Ability to block progesterone induced alkaline phosphatase activity in T47D human breast cancer cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237966(CHEMBL4078377)
Affinity DataIC50:  3.06E+3nMAssay Description:Inhibition of human IAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237924(CHEMBL4102277)
Affinity DataIC50:  3.12E+3nMAssay Description:Inhibition of human IAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237920(CHEMBL4087225)
Affinity DataIC50:  3.21E+3nMAssay Description:Displacement of [3H]dexamethasone from human Glucocorticoid receptor (GR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237928(CHEMBL4084312)
Affinity DataIC50:  3.22E+3nMAssay Description:Effect on human Glucocorticoid receptor (GR) in a whole cell assay to measure functional cellular GR-antagonism (GRAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237927(CHEMBL4086809)
Affinity DataIC50:  3.53E+3nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237941(CHEMBL4073985)
Affinity DataIC50:  3.58E+3nMAssay Description:Inhibition of human IAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237925(CHEMBL4103223)
Affinity DataIC50:  3.59E+3nMAssay Description:Inhibition of human IAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237944(CHEMBL4094013)
Affinity DataIC50:  3.69E+3nMAssay Description:Inhibition of human TNAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237947(CHEMBL4083749)
Affinity DataIC50:  3.91E+3nMAssay Description:Inhibition of human IAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237965(CHEMBL4068298)
Affinity DataIC50:  4.06E+3nMAssay Description:Inhibition of human IAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237917(CHEMBL4059741)
Affinity DataIC50:  4.06E+3nMAssay Description:Ability to block progesterone induced alkaline phosphatase activity in T47D human breast cancer cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237921(CHEMBL4065375)
Affinity DataIC50:  4.18E+3nMAssay Description:Displacement of [3H]dexamethasone from human Glucocorticoid receptor (GR); Value ranges from 1273-2947 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237939(CHEMBL4077330)
Affinity DataIC50:  4.57E+3nMAssay Description:Inhibition of human IAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237929(CHEMBL4082634)
Affinity DataIC50:  4.63E+3nMAssay Description:Inhibition of human IAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237943(CHEMBL4086241)
Affinity DataIC50:  4.65E+3nMAssay Description:Inhibition of human IAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237913(CHEMBL4091160)
Affinity DataIC50:  5.16E+3nMAssay Description:Inhibition of human IAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237962(CHEMBL4079164)
Affinity DataIC50:  5.49E+3nMAssay Description:Inhibition of human IAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237960(CHEMBL4103132)
Affinity DataIC50:  5.52E+3nMAssay Description:Inhibition of human IAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237919(CHEMBL4101742)
Affinity DataIC50:  5.95E+3nMAssay Description:Agonistic activity measures the ability to induce alkaline phosphatase in T47D human breast cancer cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50237961(CHEMBL4060753)
Affinity DataIC50:  6.29E+3nMAssay Description:Inhibition of human IAP using CDP-star as substrate pretreated for 10 mins followed by substrate addition measured after 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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