Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 8026
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [1-140](Homo sapiens (Human))
The University Of Queensland

LigandPNGBDBM228836(LQEEWETVM | PTHRct-9)
Affinity DataKi:  1.40E+3nM ΔG°:  -33.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [133-300](Homo sapiens (Human))
The University Of Queensland

LigandPNGBDBM228839(b-PTHRct-22 | biotin-DEEASCPERPPALLQEEWETVM)
Affinity DataKi:  7.00E+3nM ΔG°:  -29.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [1-140](Homo sapiens (Human))
The University Of Queensland

LigandPNGBDBM228838(Cys-PTHRct-9 | LQEEWECVM)
Affinity DataKi:  1.10E+4nM ΔG°:  -28.1kJ/molepH: 7.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [1-140](Homo sapiens (Human))
The University Of Queensland

LigandPNGBDBM228837(LQEEWETVM (phosphorylated Thr) | PTHR-p-Thrct-9)
Affinity DataKi:  1.21E+5nM ΔG°:  -22.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [1-140](Homo sapiens (Human))
The University Of Queensland

LigandPNGBDBM228845(FITC-LQEEWETVM | FITC-PTHRct9)
Affinity DataKd:  400nMpH: 6.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [133-300](Homo sapiens (Human))
The University Of Queensland

LigandPNGBDBM228845(FITC-LQEEWETVM | FITC-PTHRct9)
Affinity DataKd:  400nMpH: 6.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [1-140](Homo sapiens (Human))
The University Of Queensland

LigandPNGBDBM228845(FITC-LQEEWETVM | FITC-PTHRct9)
Affinity DataKd:  1.00E+3nMpH: 7.0 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [133-300](Homo sapiens (Human))
The University Of Queensland

LigandPNGBDBM228845(FITC-LQEEWETVM | FITC-PTHRct9)
Affinity DataKd:  600nMpH: 7.0 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [1-140](Homo sapiens (Human))
The University Of Queensland

LigandPNGBDBM228845(FITC-LQEEWETVM | FITC-PTHRct9)
Affinity DataKd:  1.00E+3nMpH: 7.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [133-300](Homo sapiens (Human))
The University Of Queensland

LigandPNGBDBM228845(FITC-LQEEWETVM | FITC-PTHRct9)
Affinity DataKd:  600nMpH: 7.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [1-140](Homo sapiens (Human))
The University Of Queensland

LigandPNGBDBM228845(FITC-LQEEWETVM | FITC-PTHRct9)
Affinity DataKd:  4.70E+3nMpH: 7.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [133-300](Homo sapiens (Human))
The University Of Queensland

LigandPNGBDBM228845(FITC-LQEEWETVM | FITC-PTHRct9)
Affinity DataKd:  2.40E+3nMpH: 7.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [1-140](Homo sapiens (Human))
The University Of Queensland

LigandPNGBDBM228839(b-PTHRct-22 | biotin-DEEASCPERPPALLQEEWETVM)
Affinity DataKd:  1.60E+4nMpH: 7.4 T: 2°CAssay Description:SPR measurements were performed with a Biacore X100 instrument (GE Healthcare Life Sciences, Piscataway, NJ) at 15.0 °C. The biotinylated PTHRct-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [133-300](Homo sapiens (Human))
The University Of Queensland

LigandPNGBDBM228840(PTHRct-8 | QEEWETVM)
Affinity DataKd:  9.70E+3nMpH: 8.0 T: 2°CAssay Description:ITC measurements were conducted on a Microcal iTC200 (Malvern Instruments) in buffer consisting of 25 mM Tris (pH 8.0) and 100 mM NaCl. Proteins were...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [1-140](Homo sapiens (Human))
The University Of Queensland

LigandPNGBDBM228840(PTHRct-8 | QEEWETVM)
Affinity DataKd:  1.17E+4nMpH: 8.0 T: 2°CAssay Description:ITC measurements were conducted on a Microcal iTC200 (Malvern Instruments) in buffer consisting of 25 mM Tris (pH 8.0) and 100 mM NaCl. Proteins were...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [133-300](Homo sapiens (Human))
The University Of Queensland

LigandPNGBDBM228839(b-PTHRct-22 | biotin-DEEASCPERPPALLQEEWETVM)
Affinity DataKd:  1.15E+4nMpH: 7.4 T: 2°CAssay Description:SPR measurements were performed with a Biacore X100 instrument (GE Healthcare Life Sciences, Piscataway, NJ) at 15.0 °C. The biotinylated PTHRct-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed