Compile Data Set for Download or QSAR
maximum 50k data
Found 71 Enz. Inhib. hit(s) with all data for entry = 50001331
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276535(CHEMBL4169732)
Affinity DataIC50:  750nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276462(CHEMBL4171638)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276597(CHEMBL4165670)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276547(CHEMBL4175880)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276426(CHEMBL4162248)
Affinity DataIC50:  1.22E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276521(CHEMBL4159529)
Affinity DataIC50:  1.32E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276527(CHEMBL4166108)
Affinity DataIC50:  1.42E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276529(CHEMBL4176308)
Affinity DataIC50:  1.45E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276518(CHEMBL4166139)
Affinity DataIC50:  1.76E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276503(CHEMBL4164439)
Affinity DataIC50:  1.99E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276452(CHEMBL4159319)
Affinity DataIC50:  2.03E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276523(CHEMBL4163296)
Affinity DataIC50:  2.11E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276504(CHEMBL4162713)
Affinity DataIC50:  2.24E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276424(CHEMBL4169565)
Affinity DataIC50:  2.42E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276526(CHEMBL4164401)
Affinity DataIC50:  2.56E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276468(CHEMBL4162887)
Affinity DataIC50:  2.66E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276541(CHEMBL4168679)
Affinity DataIC50:  2.74E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276524(CHEMBL4166740)
Affinity DataIC50:  2.87E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276382(CHEMBL4176515)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276415(CHEMBL4165448)
Affinity DataIC50:  3.05E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276502(CHEMBL4161033)
Affinity DataIC50:  3.56E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276544(CHEMBL4164153)
Affinity DataIC50:  3.75E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276594(CHEMBL4177413)
Affinity DataIC50:  4.01E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276477(CHEMBL4174447)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276505(CHEMBL4164202)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276469(CHEMBL4174641)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276533(CHEMBL4169336)
Affinity DataIC50:  5.17E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276419(CHEMBL4170150)
Affinity DataIC50:  5.39E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276543(CHEMBL4172029)
Affinity DataIC50:  5.53E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276596(CHEMBL4175078)
Affinity DataIC50:  5.74E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276470(CHEMBL4177388)
Affinity DataIC50:  6.27E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276429(CHEMBL4174219)
Affinity DataIC50:  6.65E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276536(CHEMBL4159073)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276550(CHEMBL4160931)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276476(CHEMBL4165907)
Affinity DataIC50:  7.77E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276430(CHEMBL4161825)
Affinity DataIC50:  8.14E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276534(CHEMBL4173146)
Affinity DataIC50:  8.16E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276584(CHEMBL4167226)
Affinity DataIC50:  8.46E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276595(CHEMBL4171200)
Affinity DataIC50:  8.77E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276422(CHEMBL4171229)
Affinity DataIC50:  8.92E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276532(CHEMBL4174421)
Affinity DataIC50:  9.17E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276514(CHEMBL4162687)
Affinity DataIC50:  9.65E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276478(CHEMBL4163775)
Affinity DataIC50:  9.68E+3nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276583(CHEMBL4172227)
Affinity DataIC50:  1.16E+4nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276549(CHEMBL4176055)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276404(CHEMBL4160759)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276425(CHEMBL4169526)
Affinity DataIC50:  1.38E+4nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276525(CHEMBL4175052)
Affinity DataIC50:  1.48E+4nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276522(CHEMBL4173605)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50276433(CHEMBL4173590)
Affinity DataIC50:  1.51E+4nMAssay Description:Inhibition of perforin (unknown origin)-mediated 51Cr-labelled human Jurkat cell lysis preincubated with protein for 30 mins followed by cell additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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