Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50000795
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50260459(CHEMBL4099907)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of p97 (unknown origin) expressed in Escherichia coli BL21(DE3) preincubated for 10 mins followed by ATP addition measured after 60 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX39A(Homo sapiens)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50260460(ELISABATIN A)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of DDX39A (unknown origin) expressed in Escherichia coli BL21(Rosetta 2) preincubated for 10 mins followed by ATP addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable ATP-dependent RNA helicase DDX17(Homo sapiens)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50260460(ELISABATIN A)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of DDX17 (unknown origin) expressed in Escherichia coli BL21(DE3) preincubated for 10 mins followed by ATP addition measured after 120 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable ATP-dependent RNA helicase DDX17(Homo sapiens)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50260459(CHEMBL4099907)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of DDX17 (unknown origin) expressed in Escherichia coli BL21(DE3) preincubated for 10 mins followed by ATP addition measured after 120 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50260460(ELISABATIN A)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of DDX3 (unknown origin) preincubated for 10 mins followed by ATP addition by malachite green dye-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX39A(Homo sapiens)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50260459(CHEMBL4099907)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of DDX39A (unknown origin) expressed in Escherichia coli BL21(Rosetta 2) preincubated for 10 mins followed by ATP addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target60 kDa heat shock protein, mitochondrial(Homo sapiens)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50260459(CHEMBL4099907)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GroEL (unknown origin) expressed in Escherichia coli DH5 alpha preincubated for 10 mins followed by ATP addition by malachite green dye...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock 70 kDa protein 1A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50260460(ELISABATIN A)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HSPA1A (unknown origin) expressed in Escherichia coli BL21(DE3) preincubated for 10 mins followed by ATP addition by malachite green dy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock 70 kDa protein 1A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50260459(CHEMBL4099907)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HSPA1A (unknown origin) expressed in Escherichia coli BL21(DE3) preincubated for 10 mins followed by ATP addition by malachite green dy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50260459(CHEMBL4099907)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of DDX3 (unknown origin) preincubated for 10 mins followed by ATP addition by malachite green dye-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50260460(ELISABATIN A)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of p97 (unknown origin) expressed in Escherichia coli BL21(DE3) preincubated for 10 mins followed by ATP addition measured after 60 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target60 kDa heat shock protein, mitochondrial(Homo sapiens)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50260460(ELISABATIN A)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GroEL (unknown origin) expressed in Escherichia coli DH5 alpha preincubated for 10 mins followed by ATP addition by malachite green dye...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed