Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50002936
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50464950(CHEMBL4277084)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50464949(CHEMBL4288827)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50464952(CHEMBL4290873)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50464954(CHEMBL4290458)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50464957(CHEMBL4291770)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50464948(CHEMBL4069395)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50464956(CHEMBL4280239)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50464951(CHEMBL4294266)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50464953(CHEMBL4282585)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50464955(CHEMBL4292234)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed