Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50008331
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50518208(CHEMBL4592897)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of recombinant human N-terminal poly histidine-tagged PTP1B (Glu2 to Asn321 residues) expressed in Escherichia coli using pNPP as substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50518208(CHEMBL4592897)
Affinity DataKd:  8.40nMAssay Description:Binding affinity to recombinant human N-terminal poly histidine-tagged PTP1B (Glu2 to Asn321 residues) expressed in Escherichia coli by surface plasm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50518206(CHEMBL4557598)
Affinity DataKd:  27nMAssay Description:Binding affinity to recombinant human N-terminal poly histidine-tagged PTP1B (Glu2 to Asn321 residues) expressed in Escherichia coli by surface plasm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50518207(CHEMBL4446033)
Affinity DataKd:  128nMAssay Description:Binding affinity to recombinant human N-terminal poly histidine-tagged PTP1B (Glu2 to Asn321 residues) expressed in Escherichia coli by surface plasm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed