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Found 11 Enz. Inhib. hit(s) with all data for entry = 50006846
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50069985((S)-4-methyl-2-(3-phenyl-propionylamino)-pentanoic...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of chymotrypsin like activity of 26S proteasome beta 5 subunit (unknown origin) by fluorescence assayMore data for this Ligand-Target Pair
TargetCalpain-2 catalytic subunit(Sus scrofa)
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50503849(CHEMBL4590466)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant porcine calpain 2 protease using BODIPY-FL casein as substrate measured at 30 secs time interval for 30 mins by fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50503846(CHEMBL4540394)
Affinity DataIC50:  27nMAssay Description:Inhibition of recombinant porcine calpain 2 protease using BODIPY-FL casein as substrate measured at 30 secs time interval for 30 mins by fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50503847(CHEMBL4574306)
Affinity DataIC50:  34nMAssay Description:Inhibition of recombinant porcine calpain 2 protease using BODIPY-FL casein as substrate measured at 30 secs time interval for 30 mins by fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50503849(CHEMBL4590466)
Affinity DataIC50:  139nMAssay Description:Inhibition of chymotrypsin like activity of 26S proteasome beta 5 subunit (unknown origin) by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50503845(CHEMBL4531762)
Affinity DataIC50:  160nMAssay Description:Inhibition of recombinant porcine calpain 2 protease using BODIPY-FL casein as substrate measured at 30 secs time interval for 30 mins by fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50503847(CHEMBL4574306)
Affinity DataIC50:  189nMAssay Description:Inhibition of chymotrypsin like activity of 26S proteasome beta 5 subunit (unknown origin) by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50503848(CHEMBL4475662)
Affinity DataIC50:  220nMAssay Description:Inhibition of chymotrypsin like activity of 26S proteasome beta 5 subunit (unknown origin) by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50503845(CHEMBL4531762)
Affinity DataIC50:  269nMAssay Description:Inhibition of chymotrypsin like activity of 26S proteasome beta 5 subunit (unknown origin) by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50503846(CHEMBL4540394)
Affinity DataIC50:  514nMAssay Description:Inhibition of chymotrypsin like activity of 26S proteasome beta 5 subunit (unknown origin) by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50503848(CHEMBL4475662)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of recombinant porcine calpain 2 protease using BODIPY-FL casein as substrate measured at 30 secs time interval for 30 mins by fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed