TargetHistamine H3 receptor(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Inhibition of human histamine H3 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]-LSD from recombinant human 5HT6 receptor expressed in CHOK1 cells measured after 60 mins by microbeta scintillation counting met...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Inhibition of human histamine H3 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 76nMAssay Description:Inhibition of human histamine H3 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 84nMAssay Description:Inhibition of human histamine H3 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 128nMAssay Description:Inhibition of human histamine H3 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 240nMAssay Description:Displacement of [3H]-LSD from recombinant human 5HT6 receptor expressed in CHOK1 cells measured after 60 mins by microbeta scintillation counting met...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 2.50E+3nMAssay Description:Inhibition of human histamine H3 receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 3.53E+4nMAssay Description:Inhibition of alpha4beta2 nAChR (unknown origin)More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 6.68E+4nMAssay Description:Inhibition of alpha7 nAChR (unknown origin)More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human MAOAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of COX2 in lympho-monocytes (unknown origin) preincubated for 30 mins followed by LPS challenged measured after 24 hrs by EIAMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 15.8nMAssay Description:Inhibition of 5HTT (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured aft...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Inhibition of rat AChEMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:Inhibition of human MAOBMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human MAOBMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 145nMAssay Description:Inhibition of human MAOAMore data for this Ligand-Target Pair
Affinity DataIC50: 196nMAssay Description:Inhibition of recombinant human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured aft...More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of human BChEMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of COX2 in lympho-monocytes (unknown origin) preincubated for 30 mins followed by LPS challenged measured after 24 hrs by EIAMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of human BChEMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of MOR (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 810nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of TRPV1 (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
Affinity DataIC50: 1.69E+3nMAssay Description:Inhibition of human BChEMore data for this Ligand-Target Pair
Affinity DataIC50: 1.82E+3nMAssay Description:Inhibition of human BChEMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human MAOBMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of M1R (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
TargetCarboxylic ester hydrolase(Rattus norvegicus (rat))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of rat BChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of electric eel AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of ovine COX2More data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of equine BChEMore data for this Ligand-Target Pair
TargetMonoglyceride lipase(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of FAAH (unknown origin)More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 1.14E+4nMAssay Description:Inhibition of human MAOAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of COX1 in human platelets after 30 mins by mass spectrometry analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 1.45E+4nMAssay Description:Inhibition of human alpha7 nAChR expressed in Xenopus laevis oocytes at -60 mV holding potential by two-electrode voltage-clamp techniqueMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 1.61E+4nMAssay Description:Inhibition of COX1 in human platelets after 30 mins by mass spectrometry analysisMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 1.62E+4nMAssay Description:Inhibition of ovine COX1More data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of BACE1 (unknown origin) using EVNLDAEF as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.73E+4nMAssay Description:Inhibition of human BChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 8.61E+4nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair