Found 108 Enz. Inhib. hit(s) with all data for entry = 50008488 
Affinity DataKi: 4.80nMAssay Description:Displacement of [3H]SR141716A from human CB1R receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Displacement of [3H]SR141716A from human CB1R receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
Affinity DataKi: 88nMAssay Description:Displacement of [3H]CP55940 from human CB1R receptor expressed in CHO cell membranes after 60 mins by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
Affinity DataKi: 94nMAssay Description:Displacement of [3H]CP55940 from human CB1R receptor expressed in CHO cell membranes after 60 mins by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Displacement of [3H]CP55940 from human CB1R receptor expressed in CHO cell membranes after 60 mins by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Displacement of [3H]CP55940 from human CB1R receptor expressed in CHO cell membranes after 60 mins by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Displacement of [3H]SR141716A from human CB1R receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.30E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1R receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 700nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced inhibition of forskolin-stimu...More data for this Ligand-Target Pair
Affinity DataEC50: 750nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+3nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: 26nMAssay Description:Allosteric agonist activity at N-terminal GFP-tagged rat CB1R expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP production a...More data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Positive allosteric modulatory activity at N-terminal GFP-tagged rat CB1R receptor expressed in HEK293 cells assessed as CP55940 EC50 for inhibition ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.70nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced inhibition of forskolin-induc...More data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:Positive allosteric modulatory activity at N-terminal GFP-tagged rat CB1R receptor expressed in HEK293 cells assessed as CP55940 EC50 for inhibition ...More data for this Ligand-Target Pair
Affinity DataEC50: 9.10nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced inhibition of forskolin-stimu...More data for this Ligand-Target Pair
Affinity DataEC50: 710nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: 47nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cell membranes assessed as increase in G-protein coupling by measuring [35S]GTPgammaS binding...More data for this Ligand-Target Pair
Affinity DataEC50: 940nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: 900nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: 740nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: 1.15E+3nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced inhibition of forskolin-stimu...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: 750nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: 260nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced inhibition of forskolin-stimu...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced inhibition of forskolin-stimu...More data for this Ligand-Target Pair
Affinity DataEC50: 21nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced inhibition of forskolin-stimu...More data for this Ligand-Target Pair
Affinity DataEC50: 28nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced inhibition of forskolin-stimu...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: 2.10E+3nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: 510nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: 1.14E+3nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: 3.10E+3nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced inhibition of forskolin-stimu...More data for this Ligand-Target Pair
Affinity DataEC50: 230nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced inhibition of forskolin-stimu...More data for this Ligand-Target Pair
Affinity DataEC50: 191nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced inhibition of forskolin-stimu...More data for this Ligand-Target Pair
Affinity DataEC50: 4.00E+3nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+3nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: 2.50E+3nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+3nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced inhibition of forskolin-stimu...More data for this Ligand-Target Pair
Affinity DataEC50: 230nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced inhibition of forskolin-stimu...More data for this Ligand-Target Pair
Affinity DataEC50: 690nMAssay Description:Allosteric agonist activity at N-terminal GFP-tagged rat CB1R expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP production a...More data for this Ligand-Target Pair
Affinity DataEC50: 240nMAssay Description:Allosteric agonist activity at N-terminal GFP-tagged rat CB1R expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP production a...More data for this Ligand-Target Pair
Affinity DataEC50: 27nMAssay Description:Allosteric agonist activity at N-terminal GFP-tagged rat CB1R expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP production a...More data for this Ligand-Target Pair
Affinity DataEC50: 4.30nMAssay Description:Allosteric agonist activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 90 mins by hi...More data for this Ligand-Target Pair
Affinity DataEC50: 3.90nMAssay Description:Allosteric agonist activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 90 mins by hi...More data for this Ligand-Target Pair
Affinity DataEC50: 8.10nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced inhibition of forskolin-induc...More data for this Ligand-Target Pair
Affinity DataEC50: 2.20nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced inhibition of forskolin-induc...More data for this Ligand-Target Pair
