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Found 15 Enz. Inhib. hit(s) with all data for entry = 50010633
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataKi:  13nMAssay Description:Mixed type inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50540764(CHEMBL4648322)
Affinity DataKi:  19nMAssay Description:Mixed type inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50424045(CHEMBL2314726)
Affinity DataKi:  93nMAssay Description:Mixed type inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50424045(CHEMBL2314726)
Affinity DataKi:  93.4nMAssay Description:Mixed type inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50540764(CHEMBL4648322)
Affinity DataIC50:  19nMAssay Description:Inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50540765(CHEMBL4639105)
Affinity DataIC50:  181nMAssay Description:Inhibition of human BChE using butyrylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50540766(CHEMBL4646080)
Affinity DataIC50:  223nMAssay Description:Inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50424045(CHEMBL2314726)
Affinity DataIC50:  380nMAssay Description:Inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50424045(CHEMBL2314726)
Affinity DataIC50:  380nMAssay Description:Inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50540765(CHEMBL4639105)
Affinity DataIC50:  748nMAssay Description:Inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50424045(CHEMBL2314726)
Affinity DataIC50:  2.33E+3nMAssay Description:Inhibition of human BChE using butyrylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50424045(CHEMBL2314726)
Affinity DataIC50:  2.33E+3nMAssay Description:Inhibition of human BChE using butyrylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of human BChE using butyrylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50540764(CHEMBL4648322)
Affinity DataIC50:  1.41E+4nMAssay Description:Inhibition of human BChE using butyrylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed