Compile Data Set for Download or QSAR
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Found 21 Enz. Inhib. hit(s) with all data for entry = 50029949
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50017721(1-Methyl-4-(5H-dibenzo(a,d)cycloheptenylidene)pipe...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289607(4,6-Di-furan-3-yl-2-(4-methyl-piperazin-1-yl)-pyri...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289603(2-(4-Methyl-piperazin-1-yl)-4,6-di-thiophen-2-yl-p...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289609(4-Furan-3-yl-2-(4-methyl-piperazin-1-yl)-6-phenyl-...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289608(4-Furan-3-yl-2-(4-methyl-piperazin-1-yl)-pyrimidin...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289602(4-Furan-3-yl-2-(4-methyl-piperazin-1-yl)-6-thiophe...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289605(4-Furan-2-yl-6-furan-3-yl-2-(4-methyl-piperazin-1-...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289601(4-Furan-3-yl-6-methyl-2-(4-methyl-piperazin-1-yl)-...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289606(2-(4-Methyl-piperazin-1-yl)-4-thiophen-2-yl-pyrimi...)
Affinity DataKi:  208nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289601(4-Furan-3-yl-6-methyl-2-(4-methyl-piperazin-1-yl)-...)
Affinity DataKi:  265nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289605(4-Furan-2-yl-6-furan-3-yl-2-(4-methyl-piperazin-1-...)
Affinity DataKi:  415nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289606(2-(4-Methyl-piperazin-1-yl)-4-thiophen-2-yl-pyrimi...)
Affinity DataKi:  484nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289600(2-(4-Methyl-piperazin-1-yl)-4-phenyl-pyrimidine | ...)
Affinity DataKi:  613nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289607(4,6-Di-furan-3-yl-2-(4-methyl-piperazin-1-yl)-pyri...)
Affinity DataKi:  621nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289608(4-Furan-3-yl-2-(4-methyl-piperazin-1-yl)-pyrimidin...)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289604(4-Furan-2-yl-2-(4-methyl-piperazin-1-yl)-pyrimidin...)
Affinity DataKi:  745nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289604(4-Furan-2-yl-2-(4-methyl-piperazin-1-yl)-pyrimidin...)
Affinity DataKi:  810nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289603(2-(4-Methyl-piperazin-1-yl)-4,6-di-thiophen-2-yl-p...)
Affinity DataKi:  972nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289609(4-Furan-3-yl-2-(4-methyl-piperazin-1-yl)-6-phenyl-...)
Affinity DataKi:  1.34E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289600(2-(4-Methyl-piperazin-1-yl)-4-phenyl-pyrimidine | ...)
Affinity DataKi:  2.10E+3nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289602(4-Furan-3-yl-2-(4-methyl-piperazin-1-yl)-6-thiophe...)
Affinity DataKi:  2.24E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article