Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50029951
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50099216((2S,3S)-1-[2-(3-Benzyloxycarbonyl-phenyl)-acetyl]-...)
Affinity DataIC50:  226nMAssay Description:Concentration required for inhibition of 50% of the cleavage of para-nitroanilide from MeO-Suc-Arg-Pro-Tyr-pNA.HCl by Prostate specific antigen PSAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50099216((2S,3S)-1-[2-(3-Benzyloxycarbonyl-phenyl)-acetyl]-...)
Affinity DataIC50:  226nMAssay Description:Concentration required for inhibition of 50% of the cleavage of para-nitroanilide from MeO-Suc-Arg-Pro-Tyr-pNA.HCl by Prostate specific antigen PSAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289630((2S,3S)-3-Benzyl-1-[2-(3-carboxy-phenyl)-acetyl]-4...)
Affinity DataIC50:  1.34E+3nMAssay Description:Concentration required for inhibition of 50% of the cleavage of para-nitroanilide from MeO-Suc-Arg-Pro-Tyr-pNA.HCl by Prostate specific antigen PSAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50099218((2S,3S)-3-Benzyl-1-[2-(3-benzyloxycarbonyl-phenyl)...)
Affinity DataIC50:  1.43E+3nMAssay Description:Concentration required for inhibition of 50% of the cleavage of para-nitroanilide from MeO-Suc-Arg-Pro-Tyr-pNA.HCl by Prostate specific antigen PSAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50099221((2S,3S)-1-[2-(3-Benzyloxycarbonyl-phenyl)-acetyl]-...)
Affinity DataIC50:  3.50E+3nMAssay Description:Concentration required for inhibition of 50% of the cleavage of para-nitroanilide from MeO-Suc-Arg-Pro-Tyr-pNA.HCl by Prostate specific antigen PSAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50099213((2S,3S)-3-Benzyl-1-{2-[3-(4-carboxy-benzyloxycarbo...)
Affinity DataIC50:  5.84E+3nMAssay Description:Concentration required for inhibition of 50% of the cleavage of para-nitroanilide from MeO-Suc-Arg-Pro-Tyr-pNA.HCl by Prostate specific antigen PSAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50099205((2S,3S)-3-Benzyl-1-[2-(3-benzyloxycarbonyl-phenyl)...)
Affinity DataIC50:  8.98E+3nMAssay Description:Concentration required for inhibition of 50% of the cleavage of para-nitroanilide from MeO-Suc-Arg-Pro-Tyr-pNA.HCl by Prostate specific antigen PSAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50099208((2S,3S)-3-Benzyl-1-[2-(3-carboxy-phenyl)-acetyl]-4...)
Affinity DataIC50: >3.00E+4nMAssay Description:Concentration required for inhibition of 50% of the cleavage of para-nitroanilide from MeO-Suc-Arg-Pro-Tyr-pNA.HCl by Prostate specific antigen PSAMore data for this Ligand-Target Pair
In DepthDetails Article