Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50003461
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Monash University

Curated by ChEMBL
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  5.50E+3nMAssay Description:Affinity pKi for 5-hydroxytryptamine 2C receptor was measured in rat cortex homogenates.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  5.62E+3nMAssay Description:Affinity pKi for Alpha-2 adrenergic receptor was measured in rat cortex homogenates.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Monash University

Curated by ChEMBL
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  7.94E+3nMAssay Description:Affinity pKi for 5-hydroxytryptamine 2A receptor was measured in rat cortex homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Monash University

Curated by ChEMBL
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  9.33E+3nMAssay Description:Affinity pKi for 5-hydroxytryptamine 1A receptor was measured in rat cortex homogenates.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  1.00E+4nMAssay Description:Affinity pKi for 5-hydroxytryptamine 1D receptor was measured in calf caudate homogenateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Monash University

Curated by ChEMBL
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  1.07E+4nMAssay Description:Affinity pKi for Dopamine receptor D2 was measured in rat cortex homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Monash University

Curated by ChEMBL
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  1.12E+4nMAssay Description:Affinity pKi for Alpha-1 adrenergic receptor was measured in rat cortex homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Monash University

Curated by ChEMBL
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  3.24E+4nMAssay Description:Affinity pKi for Dopamine receptor D1 was measured in rat cortex homogenates.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))
Monash University

Curated by ChEMBL
LigandPNGBDBM50471285(CHEMBL76480)
Affinity DataKi:  4.57E+4nMAssay Description:Affinity pKi for Beta adrenergic receptor was measured in rat cortex homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed