Compile Data Set for Download or QSAR
maximum 50k data
Found 45 Enz. Inhib. hit(s) with all data for entry = 50007577
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064853(CHEMBL436961 | Y-c[D-Pen-(3-I)Tyr-GSFC]KR-NH2)
Affinity DataIC50:  130nMAssay Description:Inhibition of c-Src tyrosine kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064834(CHEMBL216490 | Y-c[D-Pen-(3,5-diI)Tyr-GSFC]KR-NH2)
Affinity DataIC50:  540nMAssay Description:Inhibition of c-Src tyrosine kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064828(CHEMBL412218 | Y-c[D-Pen-(2R,3R)-2-Me-(2')Nal-GSFC...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of c-Src tyrosine kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064836(CHEMBL384640 | Y-c[Pen-YGSFC]KR-NH2)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064843(CHEMBL414159 | Y-c[D-Pen-(2S,3S)-2-Me-(2')Nal-GSFC...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of c-Src tyrosine kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064832(CHEMBL405681 | Y-c[D-Pen-(2')Nal-GSFC]KR-NH2)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of c-Src tyrosine kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064847(CHEMBL413670 | Y-c[D-Pen-(2S,3R)-2-Me-(2')Nal-GSFC...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of c-Src tyrosine kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064838(CHEMBL267152 | Y-c[Pen-(2')Nal-GSFC]KK-NH2)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064829(CHEMBL404595 | Y-c[D-Pen-D-(2')Nal-GSFC]KR-NH2)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of c-Src tyrosine kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064848(CHEMBL408137 | Y-c[D-Pen-YGSF-D-Cys]KK-NH2)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064835((S)-6-Amino-2-((S)-6-amino-2-{[(4S,7R,10S,16S,19R,...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064846(CHEMBL266442 | Y-Pen-(2')Nal-GSFCKK-NH2)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064837(CHEMBL262212 | Y-c[D-Pen-(2R,3S)-2-Me-(2')Nal-GSFC...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of c-Src tyrosine kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064827(CHEMBL274532 | Y-c[D-Pen-YGSFC]KK-NH2 | Y-c[Pen-YG...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064827(CHEMBL274532 | Y-c[D-Pen-YGSFC]KK-NH2 | Y-c[Pen-YG...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064841(CHEMBL408655 | Y-c[D-Pen-(2')Nal-GSFC]R-NH2)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064831(CHEMBL407087 | Y-c[Pen-YGSF-D-Cys]KK-NH2)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064845(CHEMBL386921 | Y-c[Pen-YGSFC]R-NH2)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064850(CHEMBL268069 | Y-Pen-YGSFCKK-NH2)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064854(Ac-Y-c[Pen-YGSFC]KR-NH2 | CHEMBL216616)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064842(CHEMBL428640 | Y-c[Pen-YGSFC]K-NH2)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064840(CHEMBL428888 | CIYGSFCKK-NH2)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064852(CHEMBL275924 | Y-Pen-Y-D-Ala-SFCKK-NH2)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064851(Ac-c[Pen-YGSFC]KR-NH2 | CHEMBL385223)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064834(CHEMBL216490 | Y-c[D-Pen-(3,5-diI)Tyr-GSFC]KR-NH2)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of p56 Lck kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064853(CHEMBL436961 | Y-c[D-Pen-(3-I)Tyr-GSFC]KR-NH2)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of p56 Lck kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064839((4S,7R,10S,16S,19R)-19-Amino-7-benzyl-16-(4-hydrox...)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064849(CHEMBL412705 | Y-c[-Pen-Y-D-Ala-SFC]KK-NH2)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064833((4S,7R,10S,16S,19R)-19-Amino-7-benzyl-16-(4-hydrox...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064830((4S,7R,10S,16S,19R)-19-Acetylamino-7-benzyl-16-(4-...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064844(Ac-Y-c[Pen-YGSFC]KK-NH2 | CHEMBL413847)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of c-Src tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064832(CHEMBL405681 | Y-c[D-Pen-(2')Nal-GSFC]KR-NH2)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of p56 Lck kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064843(CHEMBL414159 | Y-c[D-Pen-(2S,3S)-2-Me-(2')Nal-GSFC...)
Affinity DataIC50:  2.20E+5nMAssay Description:Inhibition of p56 Lck kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064828(CHEMBL412218 | Y-c[D-Pen-(2R,3R)-2-Me-(2')Nal-GSFC...)
Affinity DataIC50:  2.60E+5nMAssay Description:Inhibition of p56 Lck kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064847(CHEMBL413670 | Y-c[D-Pen-(2S,3R)-2-Me-(2')Nal-GSFC...)
Affinity DataIC50:  2.60E+5nMAssay Description:Inhibition of p56 Lck kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064837(CHEMBL262212 | Y-c[D-Pen-(2R,3S)-2-Me-(2')Nal-GSFC...)
Affinity DataIC50:  4.70E+5nMAssay Description:Inhibition of p56 Lck kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064853(CHEMBL436961 | Y-c[D-Pen-(3-I)Tyr-GSFC]KR-NH2)
Affinity DataIC50: >8.00E+5nMAssay Description:Inhibition of Lyn kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064832(CHEMBL405681 | Y-c[D-Pen-(2')Nal-GSFC]KR-NH2)
Affinity DataIC50: >8.00E+5nMAssay Description:Inhibition of Lyn kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064834(CHEMBL216490 | Y-c[D-Pen-(3,5-diI)Tyr-GSFC]KR-NH2)
Affinity DataIC50: >8.00E+5nMAssay Description:Inhibition of Lyn kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064847(CHEMBL413670 | Y-c[D-Pen-(2S,3R)-2-Me-(2')Nal-GSFC...)
Affinity DataIC50: >8.00E+5nMAssay Description:Inhibition of Lyn kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064829(CHEMBL404595 | Y-c[D-Pen-D-(2')Nal-GSFC]KR-NH2)
Affinity DataIC50: >8.00E+5nMAssay Description:Inhibition of Lyn kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064837(CHEMBL262212 | Y-c[D-Pen-(2R,3S)-2-Me-(2')Nal-GSFC...)
Affinity DataIC50: >8.00E+5nMAssay Description:Inhibition of Lyn kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064829(CHEMBL404595 | Y-c[D-Pen-D-(2')Nal-GSFC]KR-NH2)
Affinity DataIC50: >8.00E+5nMAssay Description:Inhibition of p56 Lck kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064828(CHEMBL412218 | Y-c[D-Pen-(2R,3R)-2-Me-(2')Nal-GSFC...)
Affinity DataIC50: >8.00E+5nMAssay Description:Inhibition of Lyn kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50064843(CHEMBL414159 | Y-c[D-Pen-(2S,3S)-2-Me-(2')Nal-GSFC...)
Affinity DataIC50: >8.00E+5nMAssay Description:Inhibition of Lyn kinase against 100 uM cdc2 substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed