Compile Data Set for Download or QSAR
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Found 15 Enz. Inhib. hit(s) with all data for entry = 5888
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM98618(2-amino-1-ethyl-7-[3-hydroxy-3-(3-thienyl)but-1-yn...)
Affinity DataIC50:  2nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM98616(2-amino-1-cyclohexyl-7-(3-hydroxy-4-methoxy-3-meth...)
Affinity DataIC50:  5nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM98610(2-amino-1-ethyl-7-[3-hydroxy-3-(3-methoxyphenyl)bu...)
Affinity DataIC50:  6nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM98615(2-amino-1-ethyl-7-(3-hydroxy-3-phenyl-but-1-ynyl)-...)
Affinity DataIC50:  14nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM98608(2-amino-1-ethyl-7-[2-(1-hydroxycyclobutyl)ethynyl]...)
Affinity DataIC50:  21nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM98617(2-amino-1-ethyl-7-(3-hydroxy-4-methoxy-3-methyl-bu...)
Affinity DataIC50:  23nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM98605(2-amino-1-ethyl-7-[2-(3-hydroxytetrahydrofuran-3-y...)
Affinity DataIC50:  23nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM98611(2-amino-7-(3,4-dihydroxy-3-methyl-but-1-ynyl)-N-me...)
Affinity DataIC50:  34nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM98607(2-amino-7-(3-cyclopropyl-3-hydroxy-prop-1-ynyl)-1-...)
Affinity DataIC50:  37nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM98618(2-amino-1-ethyl-7-[3-hydroxy-3-(3-thienyl)but-1-yn...)
Affinity DataIC50:  38nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM98612(2-amino-7-(3-hydroxy-3-methyl-but-1-ynyl)-N-methyl...)
Affinity DataIC50:  40nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM98614(2-amino-7-(3,4-dihydroxy-3-methyl-but-1-ynyl)-1-et...)
Affinity DataIC50:  43nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM98606(2-amino-7-(3,4-dihydroxy-3-methyl-but-1-ynyl)-1-et...)
Affinity DataIC50:  46nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM98613(2-amino-7-(3-hydroxy-4-methoxy-3-methyl-but-1-ynyl...)
Affinity DataIC50:  65nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM98609(2-amino-7-(3-hydroxy-4-methoxy-3-methyl-but-1-ynyl...)
Affinity DataIC50:  257nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In DepthDetails US Patent