Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for entry = 5972
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM103307(US8546434, 4)
Affinity DataIC50:  0.600nMpH: 7.5 T: 2°CAssay Description:In vitro activity assay using KSP.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM34539(US8546434, 13)
Affinity DataIC50:  0.690nMAssay Description:In vitro activity assay using KSP.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM103306(US8546434, 3)
Affinity DataIC50:  0.740nMpH: 7.5 T: 2°CAssay Description:In vitro activity assay using KSP.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM103309(US8546434, 6)
Affinity DataIC50:  0.830nMpH: 7.5 T: 2°CAssay Description:In vitro activity assay using KSP.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM103305(US8546434, 2)
Affinity DataIC50:  0.830nMpH: 7.5 T: 2°CAssay Description:In vitro activity assay using KSP.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM34538(US8546434, 12)
Affinity DataIC50:  0.870nMAssay Description:In vitro activity assay using KSP.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM34536(US8546434, 10)
Affinity DataIC50:  0.900nMAssay Description:In vitro activity assay using KSP.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM103304(US8546434, 1)
Affinity DataIC50:  0.960nMpH: 7.5 T: 2°CAssay Description:In vitro activity assay using KSP.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM34532(US8546434, 7)
Affinity DataIC50:  1.23nMAssay Description:In vitro activity assay using KSP.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM34537(US8546434, 11)
Affinity DataIC50:  1.40nMAssay Description:In vitro activity assay using KSP.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM103308(US8546434, 5)
Affinity DataIC50:  1.46nMpH: 7.5 T: 2°CAssay Description:In vitro activity assay using KSP.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM34534(US8546434, 8)
Affinity DataIC50:  1.49nMAssay Description:In vitro activity assay using KSP.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM34540(US8546434, 14)
Affinity DataIC50:  2.34nMAssay Description:In vitro activity assay using KSP.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM34535(US8546434, 9)
Affinity DataIC50:  49.4nMAssay Description:In vitro activity assay using KSP.More data for this Ligand-Target Pair
In DepthDetails US Patent