Compile Data Set for Download or QSAR
maximum 50k data
Found 215 Enz. Inhib. hit(s) with all data for entry = 6408
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127166(US8791272, 2.42)
Affinity DataKi:  0.100nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM50397639(CHEMBL2181751 | US8791272, 2.47)
Affinity DataKi:  0.100nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127194(US8791272, 3.12)
Affinity DataKi:  0.100nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127191(US8791272, 3.9)
Affinity DataKi:  0.100nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127296(US8791272, 17.1)
Affinity DataKi:  0.100nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127173(US8791272, 2.50)
Affinity DataKi:  0.100nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127131(US8791272, 2.14)
Affinity DataKi:  0.200nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127104(US8791272, 1.15)
Affinity DataKi:  0.200nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127125(US8791272, 2.1)
Affinity DataKi:  0.200nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127176(US8791272, 2.53)
Affinity DataKi:  0.200nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127165(US8791272, 2.41)
Affinity DataKi:  0.200nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127164(US8791272, 2.40)
Affinity DataKi:  0.200nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127130(US8791272, 2.6)
Affinity DataKi:  0.25nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127209(US8791272, 7.5)
Affinity DataKi:  0.300nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127185(US8791272, 3.3)
Affinity DataKi:  0.300nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127161(US8791272, 2.37)
Affinity DataKi:  0.400nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127175(US8791272, 2.52)
Affinity DataKi:  0.5nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127259(US8791272, 9.27)
Affinity DataKi:  0.5nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127186(US8791272, 3.4)
Affinity DataKi:  0.5nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127138(US8791272, 2.21)
Affinity DataKi:  0.5nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127172(US8791272, 2.49)
Affinity DataKi:  0.600nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127170(US8791272, 2.46)
Affinity DataKi:  0.600nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127219(US8791272, 7.15)
Affinity DataKi:  0.600nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127189(US8791272, 3.7)
Affinity DataKi:  0.600nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127134(US8791272, 2.17)
Affinity DataKi:  0.700nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127160(US8791272, 2.36)
Affinity DataKi:  0.700nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127129(US8791272, 2.5)
Affinity DataKi:  0.75nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127212(US8791272, 7.8)
Affinity DataKi:  0.800nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127150(US8791272, 2.33)
Affinity DataKi:  0.800nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127156(US8791272, 2.10)
Affinity DataKi:  0.800nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127215(US8791272, 7.11)
Affinity DataKi:  0.900nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127245(US8791272, 9.13)
Affinity DataKi:  0.900nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127162(US8791272, 2.38)
Affinity DataKi:  1nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127221(US8791272, 7.17)
Affinity DataKi:  1.10nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127126(US8791272, 2.2)
Affinity DataKi:  1.10nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127103(US8791272, 1.14)
Affinity DataKi:  1.10nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127210(US8791272, 7.6)
Affinity DataKi:  1.20nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127157(US8791272, 2.11)
Affinity DataKi:  1.20nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127154(US8791272, 2.8)
Affinity DataKi:  1.30nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127128(US8791272, 2.4)
Affinity DataKi:  1.30nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127217(US8791272, 7.13)
Affinity DataKi:  1.30nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127132(US8791272, 2.15)
Affinity DataKi:  1.40nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127163(US8791272, 2.39)
Affinity DataKi:  1.60nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127218(US8791272, 7.14)
Affinity DataKi:  1.60nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127298(US8791272, 18.1)
Affinity DataKi:  1.60nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127155(US8791272, 2.9)
Affinity DataKi:  1.80nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127171(US8791272, 2.48)
Affinity DataKi:  1.80nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127225(US8791272, 7.21)
Affinity DataKi:  1.90nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127139(US8791272, 2.22)
Affinity DataKi:  1.90nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM127224(US8791272, 7.20)
Affinity DataKi:  2.20nMpH: 7.4Assay Description:The CRTH2 receptor binding assay is performed in a scintillation proximity assay (SPA) format with the radioligand [3H]-PGD2 (Perkin Elmer, NET616000...More data for this Ligand-Target Pair
In DepthDetails US Patent
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