Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 6663
TargetChymase(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM144347(US8969348, {4-[(1,4-Dimethyl-1H-indol-3-yl)methyl]...)
Affinity DataIC50:  7nMpH: 8.0Assay Description:Chymase assays were performed in a total volume of 15 uL in Corning black opaque 384-well microtiter plates with a non-binding surface (Corning, N.Y....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymase(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM144346(US8969348, 2-{4-[(1,4-Dimethyl-1H-indol-3-yl)methy...)
Affinity DataIC50:  9nMpH: 8.0Assay Description:Chymase assays were performed in a total volume of 15 uL in Corning black opaque 384-well microtiter plates with a non-binding surface (Corning, N.Y....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymase(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM144340(US8969348, {4-[(1,4-Dimethyl-1H-indol-3-yl)methyl]...)
Affinity DataIC50:  50nMpH: 8.0Assay Description:Chymase assays were performed in a total volume of 15 uL in Corning black opaque 384-well microtiter plates with a non-binding surface (Corning, N.Y....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymase(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM144344(US8969348, 2-[4-(Naphthalen-1-ylmethyl)-1-oxophtha...)
Affinity DataIC50:  86nMpH: 8.0Assay Description:Chymase assays were performed in a total volume of 15 uL in Corning black opaque 384-well microtiter plates with a non-binding surface (Corning, N.Y....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymase(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM144348(US8969348, 2-{4-[(1-Methyl-1H-indol-3-yl)methyl]-1...)
Affinity DataIC50:  93nMpH: 8.0Assay Description:Chymase assays were performed in a total volume of 15 uL in Corning black opaque 384-well microtiter plates with a non-binding surface (Corning, N.Y....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymase(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM144341(US8969348, [4-(Naphthalen-1-ylmethyl)-1-oxophthala...)
Affinity DataIC50:  150nMpH: 8.0Assay Description:Chymase assays were performed in a total volume of 15 uL in Corning black opaque 384-well microtiter plates with a non-binding surface (Corning, N.Y....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetChymase(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM144342(US8969348, 3-{4-[(1,4-Dimethyl-1H-indol-3-yl)methy...)
Affinity DataIC50:  160nMpH: 8.0Assay Description:Chymase assays were performed in a total volume of 15 uL in Corning black opaque 384-well microtiter plates with a non-binding surface (Corning, N.Y....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymase(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM144343(US8969348, [4-(Naphthalen-1-ylmethyl)-1-oxophthala...)
Affinity DataIC50:  170nMpH: 8.0Assay Description:Chymase assays were performed in a total volume of 15 uL in Corning black opaque 384-well microtiter plates with a non-binding surface (Corning, N.Y....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymase(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM144339(US8969348, {4-[(1-Methyl-1H-indol-3-yl)methyl]-1-o...)
Affinity DataIC50:  300nMpH: 8.0Assay Description:Chymase assays were performed in a total volume of 15 uL in Corning black opaque 384-well microtiter plates with a non-binding surface (Corning, N.Y....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymase(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM144345(US8969348, {4-[(1-Methyl-1H-indol-3-yl)methyl]-1-o...)
Affinity DataIC50:  360nMpH: 8.0Assay Description:Chymase assays were performed in a total volume of 15 uL in Corning black opaque 384-well microtiter plates with a non-binding surface (Corning, N.Y....More data for this Ligand-Target Pair
In DepthDetails US Patent