Compile Data Set for Download or QSAR
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Found 15 Enz. Inhib. hit(s) with all data for entry = 4369
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65907(2-[1-(3-chlorobenzyl)indol-3-yl]sulfonyl-N-(5-meth...)
Affinity DataEC50:  5.82E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65921(2-[1-[2-fluoro-5-(1H-pyrazol-5-yl)benzyl]indol-3-y...)
Affinity DataEC50:  3.07E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65909(CHEMBL1773100 | N-(5-methyl-1,2-oxazol-3-yl)-2-[1-...)
Affinity DataEC50:  2.19E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65910(2-[1-[(6-fluoranylpyridin-3-yl)methyl]indol-3-yl]s...)
Affinity DataEC50:  1.00E+4nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65911(2-[1-(3-chloro-2-fluoro-benzyl)indol-3-yl]sulfonyl...)
Affinity DataEC50:  5.10E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65912(2-[1-[3-(6-chloro-3-pyridyl)benzyl]indol-3-yl]sulf...)
Affinity DataEC50:  3.00E+4nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65913(2-[1-(2-chlorobenzyl)indol-3-yl]sulfonyl-N-(5-meth...)
Affinity DataEC50:  1.00E+4nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65914(2-[1-(3-bromobenzyl)indol-3-yl]sulfonyl-N-(5-methy...)
Affinity DataEC50:  3.79E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65915(N-(5-methyl-1,2-oxazol-3-yl)-2-[1-[[3-(1-methylpyr...)
Affinity DataEC50:  3.21E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65916(2-[1-(3-fluorobenzyl)indol-3-yl]sulfonyl-N-(5-meth...)
Affinity DataEC50:  5.22E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65917(2-[1-(3-bromobenzyl)-4,6-difluoro-indol-3-yl]sulfo...)
Affinity DataEC50:  5.37E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65918(2-[4,6-bis(fluoranyl)-1-[[3-(1H-pyrazol-4-yl)pheny...)
Affinity DataEC50:  1.85E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65919(2-[1-[2-fluoro-3-(1H-pyrazol-5-yl)benzyl]indol-3-y...)
Affinity DataEC50:  4.40E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65920(2-[1-(5-bromo-2-fluoro-benzyl)indol-3-yl]sulfonyl-...)
Affinity DataEC50:  1.38E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65908(2-(1-m-anisylindol-3-yl)sulfonyl-N-(5-methylisoxaz...)
Affinity DataEC50:  6.54E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay