Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 4504
TargetGeneral amino acid permease AGP1(Saccharomyces cerevisiae S288c)
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM34183(2-[4-phenyl-6-(trifluoromethyl)pyrimidin-2-yl]sulf...)
Affinity DataEC50:  4.59E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03 MH086450-01 Project Title: Chemical Screen of TOR pathway GFP fusion proteins in S. ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetGeneral amino acid permease AGP1(Saccharomyces cerevisiae S288c)
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM58019(5-methyl-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)furan-...)
Affinity DataEC50:  7.75E+5nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03 MH086450-01 Project Title: Chemical Screen of TOR pathway GFP fusion proteins in S. ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetGeneral amino acid permease AGP1(Saccharomyces cerevisiae S288c)
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM55139((4Z)-4-[[3-(4-fluorophenyl)-1-phenyl-4-pyrazolyl]m...)
Affinity DataEC50:  1.07E+6nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03 MH086450-01 Project Title: Chemical Screen of TOR pathway GFP fusion proteins in S. ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetGeneral amino acid permease AGP1(Saccharomyces cerevisiae S288c)
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM76252((6-amino-5-nitro-pyrimidin-4-yl)-(3,5-dichlorophen...)
Affinity DataEC50:  7.64E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03 MH086450-01 Project Title: Chemical Screen of TOR pathway GFP fusion proteins in S. ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay