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Found 209 Enz. Inhib. hit(s) with all data for entry = 5793
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM59558(3-(2-methyl-6-phenyl-thieno[2,3-d]pyrimidin-4-yl)s...)
Affinity DataIC50:  212nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM48242(2-[4-[(4-tert-butylbenzoyl)amino]phenyl]acetic aci...)
Affinity DataIC50:  243nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94003(3-(2-keto-4-methyl-6,7,8,9-tetrahydrobenzofuro[3,2...)
Affinity DataIC50:  276nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM38917(3-[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]pro...)
Affinity DataIC50: <300nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94046(4-(5-phenyl-1,3-oxazol-2-yl)aniline | 4-(5-phenyl-...)
Affinity DataIC50: <300nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM38998(MLS000064750 | N-(3-cyano-5,6,7,8-tetrahydro-4H-cy...)
Affinity DataIC50: <300nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM93990(3-[2-(4-chlorophenyl)-5,7-dimethyl-6-pyrazolo[1,5-...)
Affinity DataIC50:  344nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM48209(2-[4-[(3-methyl-2-furoyl)amino]phenyl]acetic acid ...)
Affinity DataIC50:  374nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94007((E)-3-[4-(2-cyanobenzyl)oxyphenyl]acrylic acid | (...)
Affinity DataIC50:  391nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94022(4-[(E)-[[4-[(2-isopropyl-5-methyl-phenoxy)methyl]b...)
Affinity DataIC50:  450nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94039(2-(2,4-Dimethyl-phenyl)-2H-benzotriazol-5-ylamine ...)
Affinity DataIC50:  452nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94053((2S)-1-[3-(2-keto-4-methyl-6,7,8,9-tetrahydrobenzo...)
Affinity DataIC50:  512nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM38964(3-[(4-methoxyphenoxy)methyl]benzoic acid | MLS0000...)
Affinity DataIC50:  781nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM93951(3-(5,7-dimethyl-2-phenyl-6-pyrazolo[1,5-a]pyrimidi...)
Affinity DataIC50:  832nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94068(MLS003120467 | N-(4-acetamidophenyl)-4-(2-methyl-3...)
Affinity DataIC50:  858nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94011((3-aminophenyl)(3,4-dimethylphenyl)methanone | (3-...)
Affinity DataIC50:  864nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM93993(4-[(4-bromo-2,5-dimethyl-pyrazole-3-carbonyl)thioc...)
Affinity DataIC50:  894nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94015(2-[4-(4-pyridin-2-ylpyrimidin-2-yl)phenoxy]acetic ...)
Affinity DataIC50:  913nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM93995(1-(3-nitrobenzyl)-1H-indole-3-carbaldehyde | 1-(3-...)
Affinity DataIC50:  978nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM59529(3-[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]-N-...)
Affinity DataIC50: <1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM87341(3-[3-(4-tert-Butyl-phenyl)-[1,2,4]oxadiazol-5-yl]-...)
Affinity DataIC50: <1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94058(3-(4-aminophenyl)-2-benzopyran-1-one | 3-(4-aminop...)
Affinity DataIC50: <1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94069(MLS001125810 | N-[[4-[(4-bromobenzoyl)amino]phenyl...)
Affinity DataIC50:  1.02E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM64363(4-[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-cycl...)
Affinity DataIC50:  1.04E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM77237(3-(5,7-dimethyl-2-phenyl-6-pyrazolo[1,5-a]pyrimidi...)
Affinity DataIC50:  1.05E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94008(3-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)sul...)
Affinity DataIC50:  1.05E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM7630(cid_2193280)
Affinity DataIC50:  1.06E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94042(2-[4-[4-(2-pyridinyl)-2-pyrimidinyl]phenoxy]acetic...)
Affinity DataIC50:  1.07E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM39089(2-(5-bromanyl-2-chloranyl-phenyl)-1,3-benzoxazol-5...)
Affinity DataIC50:  1.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM64327((5Z)-3-(2-aminoethyl)-5-(1,3-benzodioxol-5-ylmethy...)
Affinity DataIC50:  1.12E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM60223(4-methyl-N-(8-quinolinyl)benzenesulfonamide | 4-me...)
Affinity DataIC50:  1.12E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM35415(1-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-3-[2-(3-fl...)
Affinity DataIC50:  1.27E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM93958(1-[3-(5,7-dimethyl-2-phenyl-6-pyrazolo[1,5-a]pyrim...)
Affinity DataIC50:  1.39E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94054(1-[3-(2-keto-4-methyl-6,7,8,9-tetrahydrobenzofuro[...)
Affinity DataIC50:  1.41E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM93957(3-[2-(4-chlorophenyl)-5,7-dimethyl-6-pyrazolo[1,5-...)
Affinity DataIC50:  1.43E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94041((2S)-2-[3-(2-keto-4-methyl-6,7,8,9-tetrahydrobenzo...)
Affinity DataIC50:  1.61E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM93955(MLS000103529 | N-(4-acetamidophenyl)-3,5,6-trimeth...)
Affinity DataIC50:  1.64E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM36972(2-[4-[(2-isopropyl-5-methyl-phenoxy)methyl]phenyl]...)
Affinity DataIC50:  1.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM93959(3-(5,7-dimethyl-2-phenyl-6-pyrazolo[1,5-a]pyrimidi...)
Affinity DataIC50:  1.81E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM48202(4-(5-Methoxy-1H-benzoimidazol-2-yl)-phenylamine | ...)
Affinity DataIC50:  1.88E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM93967(2-[2-[(4-fluorobenzoyl)thiocarbamoylamino]thiazol-...)
Affinity DataIC50:  1.96E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94036(3-[[5-(4-chlorophenyl)-1,3,4-oxadiazol-2-yl]sulfan...)
Affinity DataIC50:  1.97E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM38983(MLS000045930 | N-(2,5-dimethoxyphenyl)-4-(5-p-phen...)
Affinity DataIC50:  1.99E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM93980(3-[(4-ethoxyphenoxy)methyl]-N'-(3-pyridinylmet...)
Affinity DataIC50:  2.03E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM48108((4-acetamidophenyl) piperidine-1-carboxylate | 1-p...)
Affinity DataIC50:  2.33E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM93968(2-[[5-(3-chloro-1-benzothiophen-2-yl)-1,3,4-oxadia...)
Affinity DataIC50:  2.36E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM93963(MLS000566332 | N-[4-[2-(2,4-dimethylphenyl)-2-keto...)
Affinity DataIC50:  2.47E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM39028(3-[(2-chloranylphenoxy)methyl]benzoic acid | 3-[(2...)
Affinity DataIC50:  2.58E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94047(2-[4-[4-(4-fluorophenyl)-2-pyrimidinyl]phenoxy]ace...)
Affinity DataIC50:  2.66E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94023(Fast Bordeaux 3B base | MLS000736833 | N-(4-amino-...)
Affinity DataIC50:  2.75E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
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