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Found 249 Enz. Inhib. hit(s) with all data for entry = 5818
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95823(MLS001220202 | N-(3-Methoxy-phenyl)-2-(8-methyl-5H...)
Affinity DataIC50:  48.3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM72157(MLS000571934 | N-[2-(1H-benzimidazol-2-yl)ethyl]-4...)
Affinity DataIC50:  170nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95868(2-[3-(2-keto-2-morpholino-acetyl)indol-1-yl]-N-[3-...)
Affinity DataIC50:  205nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95760((2S,4S)-N-(1H-benzimidazol-2-ylmethyl)-4-(4-bromop...)
Affinity DataIC50:  270nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95701(2-[4-[(6-bromanyl-1H-benzimidazol-2-yl)amino]pheny...)
Affinity DataIC50:  286nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95801((12aS)-2-methyl-6-(3-nitrophenyl)-6,7,12,12a-tetra...)
Affinity DataIC50:  393nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM74708(2-(1H-benzimidazol-2-ylmethylsulfanyl)-5-(2,4-dich...)
Affinity DataIC50:  401nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM57561(1-[1-(4-Bromo-phenyl)-2,5-dioxo-pyrrolidin-3-yl]-1...)
Affinity DataIC50:  460nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95696(MLS000121584 | N-(1,3-benzodioxol-5-yl)-2-[(8-meth...)
Affinity DataIC50:  489nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95765((2S,4S)-N-(1H-benzimidazol-2-ylmethyl)-4-(4-bromop...)
Affinity DataIC50:  498nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95798((12aS)-2-(3-hydroxypropyl)-6-(3-nitrophenyl)-6,7,1...)
Affinity DataIC50:  528nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95745(3-[4-[4-(4-acetylphenyl)-1-piperazinyl]-4-oxobutyl...)
Affinity DataIC50:  579nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95733(1-[3-[(2-methoxyphenyl)sulfamoyl]phenyl]-3-phenyl-...)
Affinity DataIC50:  644nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95793(2-[(1H-Benzoimidazol-2-ylamino)-methyl]-4,6-dichlo...)
Affinity DataIC50:  661nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95857((2S,3R,12bS)-2-((benzo[d][1,3]dioxol-5-ylmethyl)(m...)
Affinity DataIC50:  672nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95820(2-[(8-methyl-5H-[1,2,4]triazin[5,6-b]indol-3-yl)th...)
Affinity DataIC50:  720nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95811(MLS001211235 | N-(3-Bromo-phenyl)-3-[(2,4-dihydrox...)
Affinity DataIC50:  756nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM90540((3Z)-N-(4-bromophenyl)-3-(4-nitrobenzyl)oximino-pr...)
Affinity DataIC50:  784nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95818(2-(8-Fluoro-5H-[1,2,4]triazino[5,6-b]indol-3-ylsul...)
Affinity DataIC50:  785nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95761((2S,4R)-N-(1H-benzimidazol-2-ylmethyl)-4-cycloprop...)
Affinity DataIC50:  811nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95764((2S,4S)-N-(1H-benzimidazol-2-ylmethyl)-2-(4-methyl...)
Affinity DataIC50:  835nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95819(2-(8-Fluoro-5H-[1,2,4]triazino[5,6-b]indol-3-ylsul...)
Affinity DataIC50:  879nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95856((2S,3R,12bS)-2-((4-chlorobenzyl)(methyl)amino)-3-(...)
Affinity DataIC50:  974nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95800((12aS)-2-(3-isopropoxypropyl)-6-(3-nitrophenyl)-6,...)
Affinity DataIC50:  979nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95802(4-acetyl-N-[3-(trifluoromethyl)benzyl]-1H-pyrrole-...)
Affinity DataIC50:  1.16E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95831(MLS001079903 | N-[2-(4-chloroanilino)-2-keto-ethyl...)
Affinity DataIC50:  1.18E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM57346(1-[[2-(2,4-dichlorophenyl)quinolin-4-yl]carbonylam...)
Affinity DataIC50:  1.28E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95855((2S,3R,12bS)-2-((3,5-dichlorobenzyl)(methyl)amino)...)
Affinity DataIC50:  1.33E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95821(2-(8-Bromo-5H-[1,2,4]triazino[5,6-b]indol-3-ylsulf...)
Affinity DataIC50:  1.36E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95777((2S,4S)-N-(1H-benzimidazol-2-ylmethyl)-4-(1-benzot...)
Affinity DataIC50:  1.36E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95822(2-[(8-fluoranyl-5H-[1,2,4]triazino[5,6-b]indol-3-y...)
Affinity DataIC50:  1.42E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95779((2S,4S)-N-(1H-benzimidazol-2-ylmethyl)-2-[[4-(hydr...)
Affinity DataIC50:  1.47E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95739(MLS000679757 | N-(3-chloranyl-4-fluoranyl-phenyl)-...)
Affinity DataIC50:  1.47E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95810(MLS000999870 | N-(4-Methoxy-benzyl)-2-(5H-[1,2,4]t...)
Affinity DataIC50:  1.54E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM87885(MLS000700267 | S-[2-(3-methoxyanilino)-2-oxoethyl]...)
Affinity DataIC50:  1.57E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95778((2R,4R)-N-(1H-benzimidazol-2-ylmethyl)-4-(1-benzot...)
Affinity DataIC50:  1.58E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM57358(1-[[2-(3,4-dichlorophenyl)quinolin-4-yl]carbonylam...)
Affinity DataIC50:  1.64E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM76246(MLS001143266 | N-(3-bromobenzyl)-2-[(3-ethylisoxaz...)
Affinity DataIC50:  1.66E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95748((3Z)-N-(4-chlorophenyl)-3-(4-nitrobenzyl)oximino-p...)
Affinity DataIC50:  1.73E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95735(2-(1-benzimidazolyl)-N-(3-nitrophenyl)acetamide | ...)
Affinity DataIC50:  1.76E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM50869(4-(benzenesulfonyl)-N-(4-chlorophenyl)-4-[3-chloro...)
Affinity DataIC50:  1.77E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95861(2-[(3R,4S)-1-benzyl-4-(4-bromophenyl)-2-keto-pyrro...)
Affinity DataIC50:  1.78E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95799((12aS)-2-(1-benzyl-4-piperidyl)-6-(3-nitrophenyl)-...)
Affinity DataIC50:  1.82E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95766((2R,4R)-N-(1H-benzimidazol-2-ylmethyl)-4-(1,3-benz...)
Affinity DataIC50:  1.84E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95691(3-[(5-bromanylthiophen-2-yl)sulfonylamino]-N-(4-ch...)
Affinity DataIC50:  1.85E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95872(1-Nonyl-2,3,4,9-tetrahydro-1H-beta-carboline-3-car...)
Affinity DataIC50:  1.96E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95776((2R,4R)-N-(1H-benzimidazol-2-ylmethyl)-4-tert-buty...)
Affinity DataIC50:  1.99E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95825(2-[(6-bromanyl-1H-imidazo[4,5-b]pyridin-2-yl)sulfa...)
Affinity DataIC50:  2.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM71661(3-[2-(2-Methylcarbamoylmethyl-benzoimidazol-1-yl)-...)
Affinity DataIC50:  2.05E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetMethionine--tRNA ligase(Trypanosoma brucei brucei strain 927/4 GUTat10.1)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95834(MLS001143278 | N-(3-bromobenzyl)-2-[(3-methylisoxa...)
Affinity DataIC50:  2.08E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
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