Reaction Details Report a problem with these data
Target
N-formyl peptide receptor 2
Ligand
BDBM37611
Substrate
n/a
Meas. Tech.
Dose Response Assay for Formylpeptide Receptor-Like-1 (FPRL1) Ligands and Dose Response Counter-Screen Assay for Formylpeptide Receptor (FPR) Ligands
Ki
>40300±n/a nM
Comments
Extracted from aid = 520 and tid = 2
Citation
 PubChem, PC Dose Response Assay for Formylpeptide Receptor-Like-1 (FPRL1) Ligands and Dose Response Counter-Screen Assay for Formylpeptide Receptor (FPR) Ligands PubChem Bioassay (2007)[AID] 
Target
Name:
N-formyl peptide receptor 2
Synonyms:
ALXR, FPRL1, FPR2 | FMLP-related receptor I FMLP-R-I | FPR2 | FPR2_HUMAN | FPRH1 | FPRL1 | Formyl Peptide Receptor-Like 1 | HM63 | LXA4 receptor | LXA4R | Lipoxin A4 receptor | Lipoxin A4 receptor (LXA4) | RFP | hFPRL
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
38968.35
Organism:
Homo sapiens (Human)
Description:
P25090
Residue:
351
Sequence:
METNFSTPLNEYEEVSYESAGYTVLRILPLVVLGVTFVLGVLGNGLVIWVAGFRMTRTVTTICYLNLALADFSFTATLPFLIVSMAMGEKWPFGWFLCKLIHIVVDINLFGSVFLIGFIALDRCICVLHPVWAQNHRTVSLAMKVIVGPWILALVLTLPVFLFLTTVTIPNGDTYCTFNFASWGGTPEERLKVAITMLTARGIIRFVIGFSLPMSIVAICYGLIAAKIHKKGMIKSSRPLRVLTAVVASFFICWFPFQLVALLGTVWLKEMLFYGKYKIIDILVNPTSSLAFFNSCLNPMLYVFVGQDFRERLIHSLPTSLERALSEDSAPTNDTAANSASPPAETELQAM
  
Inhibitor
Name:
BDBM37611
Synonyms:
3-(furan-2-carbonyl)-4-hydroxy-1-(2-morpholin-4-ylethyl)-2-(3-prop-2-enoxyphenyl)-2H-pyrrol-5-one | 3-(furan-2-ylcarbonyl)-1-(2-morpholin-4-ylethyl)-4-oxidanyl-2-(3-prop-2-enoxyphenyl)-2H-pyrrol-5-one | 3-[2-furanyl(oxo)methyl]-4-hydroxy-1-[2-(4-morpholinyl)ethyl]-2-(3-prop-2-enoxyphenyl)-2H-pyrrol-5-one | 5-(3-Allyloxy-phenyl)-4-(furan-2-carbonyl)-3-hydroxy-1-(2-morpholin-4-yl-ethyl)-1,5-dihydro-pyrrol-2-one | 5-(3-allyloxyphenyl)-4-(2-furoyl)-3-hydroxy-1-(2-morpholinoethyl)-3-pyrrolin-2-one | MLS000034805 | SMR000013765 | cid_650032
Type:
Small organic molecule
Emp. Form.:
C24H26N2O6
Mol. Mass.:
438.473
SMILES:
C=CCOc1cccc(c1)C1C(C(=O)c2ccco2)C(=O)C(=O)N1CCN1CCOCC1
Structure:
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