Reaction Details Report a problem with these data
Target
N-formyl peptide receptor 2
Ligand
BDBM37679
Substrate
n/a
Meas. Tech.
Dose Response Assay for Formylpeptide Receptor-Like-1 (FPRL1) Ligands and Dose Response Counter-Screen Assay for Formylpeptide Receptor (FPR) Ligands
IC50
>66700±n/a nM
Comments
Extracted from aid = 520 and tid = 3
Citation
 PubChem, PC Dose Response Assay for Formylpeptide Receptor-Like-1 (FPRL1) Ligands and Dose Response Counter-Screen Assay for Formylpeptide Receptor (FPR) Ligands PubChem Bioassay (2007)[AID] 
Target
Name:
N-formyl peptide receptor 2
Synonyms:
ALXR, FPRL1, FPR2 | FMLP-related receptor I FMLP-R-I | FPR2 | FPR2_HUMAN | FPRH1 | FPRL1 | Formyl Peptide Receptor-Like 1 | HM63 | LXA4 receptor | LXA4R | Lipoxin A4 receptor | Lipoxin A4 receptor (LXA4) | RFP | hFPRL
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
38968.35
Organism:
Homo sapiens (Human)
Description:
P25090
Residue:
351
Sequence:
METNFSTPLNEYEEVSYESAGYTVLRILPLVVLGVTFVLGVLGNGLVIWVAGFRMTRTVTTICYLNLALADFSFTATLPFLIVSMAMGEKWPFGWFLCKLIHIVVDINLFGSVFLIGFIALDRCICVLHPVWAQNHRTVSLAMKVIVGPWILALVLTLPVFLFLTTVTIPNGDTYCTFNFASWGGTPEERLKVAITMLTARGIIRFVIGFSLPMSIVAICYGLIAAKIHKKGMIKSSRPLRVLTAVVASFFICWFPFQLVALLGTVWLKEMLFYGKYKIIDILVNPTSSLAFFNSCLNPMLYVFVGQDFRERLIHSLPTSLERALSEDSAPTNDTAANSASPPAETELQAM
  
Inhibitor
Name:
BDBM37679
Synonyms:
MLS000057035 | N-(1-allyl-3-cyano-pyrrolo[3,2-b]quinoxalin-2-yl)benzamide | N-(3-cyano-1-prop-2-enyl-2-pyrrolo[3,2-b]quinoxalinyl)benzamide | N-(3-cyano-1-prop-2-enyl-pyrrolo[3,2-b]quinoxalin-2-yl)benzamide | N-(3-cyano-1-prop-2-enylpyrrolo[3,2-b]quinoxalin-2-yl)benzamide | SMR000060389 | cid_2309631
Type:
Small organic molecule
Emp. Form.:
C21H15N5O
Mol. Mass.:
353.3767
SMILES:
C=CCn1c(NC(=O)c2ccccc2)c(C#N)c2nc3ccccc3nc12
Structure:
Search PDB for entries with ligand similarity: